SCHEMBL7422328

SCHEMBL7422328

CCOC(=O)CN(c1ccc([N+](=O)[O-])cc1)S(=O)(=O)c1ccccc1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.64
MAPT P10636 5/20 0.64
MEN1 O00255 4/20 0.64
ALDH1A1 P00352 4/20 0.64
HTT P42858 2/20 0.61
MAPK1 P28482 2/20 0.56
TDP1 Q9NUW8 1/20 0.56
GLA P06280 1/20 0.56
PKM P14618 1/20 0.53
NR3C1 P04150 1/20 0.53
HPGD P15428 2/20 0.51
NR1I2 O75469 1/20 0.51
RAB9A P51151 1/20 0.51
LMNA P02545 3/20 0.50
BACE1 P56817 1/20 0.50
NPSR1 Q6W5P4 1/20 0.50
RORC P51449 1/20 0.49
CA9 Q16790 1/20 0.49
KEAP1 Q14145 1/20 0.49
NFE2L2 Q16236 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5461521 0.88 PKM (0.61) KMT2AMAPTMEN1ALDH1A1HTT
SCHEMBL6608045 0.84 MAPT (0.61) KMT2AMAPTMEN1ALDH1A1HTT
SCHEMBL5624112 0.84 ALDH1A1 (0.51) KMT2AMAPTMEN1ALDH1A1MAPK1
SCHEMBL3461871 0.84 HCRTR2 (0.50) KMT2AMAPTMEN1ALDH1A1HTT
SCHEMBL7423210 0.83 ALDH1A1 (0.55) ALDH1A1MAPK1NR3C1NR1I2LMNA
SCHEMBL6574348 0.83 MMP1 (0.52) KMT2AMAPTMEN1ALDH1A1HTT
SCHEMBL28751721 0.80 ALDH1A1 (0.54) KMT2AMAPTMEN1ALDH1A1MAPK1
SCHEMBL26247562 0.80 MAPT (0.61) KMT2AMAPTMEN1ALDH1A1HTT
SCHEMBL6611414 0.80 MAPT (0.61) KMT2AMAPTMEN1ALDH1A1HTT
SCHEMBL7000752 0.80 KEAP1 (0.66) KMT2AMAPTMEN1ALDH1A1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0885205-A4 FIBRINOGEN RECEPTOR ANTAGONISTS MERCK & CO INC (US) 2002-11-27 EP disclosed
EP-0885205-A1 FIBRINOGEN RECEPTOR ANTAGONISTS Merck & Co., Inc. (US) 1998-12-23 EP disclosed
US-5780480-A THROMBOLYTIC AGENTS, ANTICOAGULANTS MERCK & CO., INC. (US) 1998-07-14 US disclosed
WO-1997031910-A1 FIBRINOGEN RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 1997-09-04 WO disclosed