SCHEMBL7423883

SCHEMBL7423883

O=C(c1cnc(Cl)nc1C(F)(F)F)N1C=C2CC=CN2Cc2ccccc21

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NFKB1 P19838 13/20 0.42
JUN P05412 2/20 0.42
NFKB2 Q00653 2/20 0.42
RELA Q04206 2/20 0.42
XPO1 O14980 4/20 0.42
ATF1 P18846 12/20 0.39
AVPR2 P30518 2/20 0.35
SCD O00767 1/20 0.34
OXTR P30559 1/20 0.33
AVPR1A P37288 1/20 0.33
HCRTR1 O43613 1/20 0.32
HCRTR2 O43614 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7419308 0.82 AVPR2 (0.44) AVPR2OXTRAVPR1AHCRTR1HCRTR2
SCHEMBL7421267 0.77 AVPR2 (0.38) AVPR2OXTRAVPR1A
SCHEMBL7421754 0.77 AVPR2 (0.50) AVPR2OXTRAVPR1A
SCHEMBL7417501 0.75 AVPR2 (0.40) AVPR2OXTRAVPR1AHCRTR1HCRTR2
SCHEMBL7420622 0.75 AVPR2 (0.43) AVPR2OXTRAVPR1A
SCHEMBL7422025 0.73 AVPR2 (0.42) AVPR2OXTRAVPR1A
SCHEMBL2313462 0.71 HSD17B3 (0.32)
SCHEMBL7549935 0.71 BCAT2 (0.34) AVPR2OXTRAVPR1A
SCHEMBL7422271 0.71 AVPR2 (0.52) AVPR2OXTRAVPR1A
SCHEMBL7424272 0.71 AVPR2 (0.50) AVPR2OXTRAVPR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1216045-A2 VASOPRESSIN AGONIST FORMULATION AND PROCESS American Cynamid Company (US) 2002-06-26 EP disclosed
WO-2001022969-A2 VASOPRESSIN AGONIST FORMULATION AND PROCESS AMERICAN CYNAMID COMPANY (US) 2001-04-05 WO disclosed
EP-1000062-A1 TRICYCLIC VASOPRESSIN AGONISTS AMERICAN HOME PRODUCTS CORPORATION (US) 2000-05-17 EP disclosed
WO-1999006409-A1 TRICYCLIC VASOPRESSIN AGONISTS AMERICAN HOME PRODUCTS CORPORATION (US) 1999-02-11 WO disclosed