SCHEMBL7424497

SCHEMBL7424497

NNc1nnc(-c2ccccc2)cc1Cc1ccccc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.41
AGTR1 P30556 1/20 0.41
SMARCA2 P51531 1/20 0.41
SMARCA4 P51532 1/20 0.41
PBRM1 Q86U86 1/20 0.41
ALDH1A1 P00352 1/20 0.39
ADORA3 P0DMS8 1/20 0.39
MAOA P21397 1/20 0.39
PTGS1 P23219 1/20 0.39
OPRM1 P35372 1/20 0.39
KCNH2 Q12809 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
BCL2 P10415 1/20 0.37
BCL2L1 Q07817 1/20 0.37
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
ACHE P22303 2/20 0.36
CYP11B1 P15538 1/20 0.36
CYP11B2 P19099 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1752856 0.81 AGTR1 (0.38) MAPTAGTR1SMARCA2SMARCA4PBRM1
SCHEMBL7438450 0.80 MAPT (0.40) MAPTAGTR1SMARCA2SMARCA4PBRM1
SCHEMBL1752842 0.76 CASP1 (0.47) SMARCA2SMARCA4PBRM1ALDH1A1BCL2
SCHEMBL14069624 0.75 SMARCA2 (0.52) MAPTAGTR1SMARCA2SMARCA4PBRM1
SCHEMBL1752808 0.73 ACHE (0.51) MAPTAGTR1SMARCA2SMARCA4PBRM1
SCHEMBL6380688 0.72 PDE4A (0.43) MAPTALDH1A1MEN1KMT2ACYP11B1
SCHEMBL1752913 0.70 MEN1 (0.54) MAPTAGTR1SMARCA2SMARCA4PBRM1
SCHEMBL1752930 0.69 MEN1 (0.44) MAPTMEN1KMT2ACYP11B1CYP11B2
SCHEMBL1752810 0.68 SMARCA2 (0.56) SMARCA2SMARCA4PBRM1MAOASMN1; SMN2
SCHEMBL1752934 0.68 NPC1 (0.49) KCNH2TDP1ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5278161-A Racemic mixtures HOFFMANN-LA ROCHE INC. (US) 1994-01-11 US disclosed
EP-0464572-A2 Aminoacid derivatives F. HOFFMANN-LA ROCHE AG (CH) 1992-01-08 EP disclosed