SCHEMBL7424982

SCHEMBL7424982

COc1ccc(CCCN2C(=O)c3ccccc3C2=O)cc1OC1CCc2ccccc21

nearest known ligand 0.53

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.51
LMNA P02545 2/20 0.48
NR1H3 Q13133 2/20 0.47
NR1H2 P55055 1/20 0.47
ABCB1 P08183 2/20 0.44
SMPD1 P17405 1/20 0.44
DRD2 P14416 1/20 0.43
PDE4A P27815 1/20 0.42
PDE4B Q07343 1/20 0.42
PDE4C Q08493 1/20 0.42
PDE4D Q08499 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11743353 0.82 ALDH1A1 (0.69) ALDH1A1LMNANR1H3NR1H2
SCHEMBL7425987 0.81 SMPD1 (0.47) ABCB1SMPD1
SCHEMBL8707317 0.80 NR1H3 (0.51) ALDH1A1LMNANR1H3NR1H2PDE4A
SCHEMBL9053567 0.77 ALDH1A1 (0.67) ALDH1A1LMNANR1H3NR1H2
SCHEMBL4637258 0.77 PDE4A (0.55) PDE4APDE4BPDE4CPDE4D
SCHEMBL8712860 0.75 QPCT (0.43) NR1H3NR1H2PDE4APDE4BPDE4C
SCHEMBL8777049 0.74 LMNA (0.72) ALDH1A1LMNANR1H3NR1H2
SCHEMBL8711619 0.73 CMA1 (0.42) ALDH1A1PDE4APDE4BPDE4CPDE4D
SCHEMBL8708949 0.73 HTR2C (0.46) ALDH1A1
SCHEMBL8711349 0.73 HTR2C (0.46) ALDH1A1NR1H3NR1H2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0874819-A1 IMIDES AS PDE III, PDE IV AND TNF INHIBITORS CELGENE CORPORATION (US) 1998-11-04 EP disclosed
WO-1997023457-A1 IMIDES AS PDE III, PDE IV AND TNF INHIBITORS CELGENE CORPORATION (US) 1997-07-03 WO disclosed