SCHEMBL7425178

SCHEMBL7425178

COC[C@H](NC(=O)C(F)(F)C(=O)C(Cc1ccc(OCc2ccccc2)cc1)NC(=O)[C@@H](NC(=O)OCc1cccnc1)C(C)C)C(C)C

nearest known ligand 0.45

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GPR132 Q9UNW8 3/20 0.44
CTSL P07711 2/20 0.43
CTSB P07858 1/20 0.43
CTSD P07339 3/20 0.42
ELANE P08246 2/20 0.42
ACACB O00763 1/20 0.42
CYP3A4 P08684 3/20 0.41
ITGB3 P05106 1/20 0.41
ITGA2B P08514 1/20 0.41
CTSS P25774 1/20 0.41
CTSK P43235 1/20 0.41
ALDH1A1 P00352 1/20 0.41
TSHR P16473 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7421246 0.96 GPR132 (0.44) GPR132CTSLCTSBCTSDELANE
SCHEMBL7417968 0.96 GPR132 (0.44) GPR132CTSLCTSBCTSDELANE
SCHEMBL7421382 0.91 REN (0.42) GPR132CTSLCTSBCTSDELANE
SCHEMBL7418157 0.90 REN (0.45) CTSDELANEITGB3ITGA2B
SCHEMBL7415239 0.89 REN (0.41) GPR132CTSLCTSBCTSDELANE
SCHEMBL8945566 0.89 CTSD (0.47) CTSBCTSDITGB3ITGA2BCTSS
SCHEMBL7933938 0.89 CTSD (0.47) CTSBCTSDITGB3ITGA2BCTSS
SCHEMBL7422064 0.88 CTSD (0.47) GPR132CTSDELANEACACBCYP3A4
SCHEMBL7421155 0.87 CTSD (0.43) CTSDITGB3ITGA2BCTSSCTSK
SCHEMBL7422846 0.86 CTSD (0.44) CTSDITGB3ITGA2BCTSSCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0773926-A1 DIFLUOROSTATONE ANTIVIRAL AGENTS MERRELL PHARMACEUTICALS INC. (US) 1997-05-21 EP claimed
WO-1996002499-A1 DIFLUOROSTATONE ANTIVIRAL AGENTS MERRELL PHARMACEUTICALS INC. (US) 1996-02-01 WO claimed
WO-1996002499-A1 DIFLUOROSTATONE ANTIVIRAL AGENTS MERRELL PHARMACEUTICALS INC. (US) 1996-02-01 WO disclosed