SCHEMBL7425294

SCHEMBL7425294

CC(C)CC(NCC(C(=O)O)c1ccccc1OCc1csc2ccc(Cl)cc12)C(=O)O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.41
KEAP1 Q14145 1/20 0.41
NFE2L2 Q16236 1/20 0.41
FFAR4 Q5NUL3 1/20 0.38
EGFR P00533 1/20 0.36
ERBB2 P04626 1/20 0.36
EPHA2 P29317 1/20 0.36
KDR P35968 1/20 0.36
EPHB4 P54760 1/20 0.36
PKM P14618 1/20 0.36
CPB1 P15086 1/20 0.36
PDCD1 Q15116 1/20 0.36
CD274 Q9NZQ7 1/20 0.36
MAPK1 P28482 1/20 0.35
EPHX1 P07099 1/20 0.35
CMA1 P23946 1/20 0.35
NTSR1 P30989 2/20 0.34
CYP2A6 P11509 1/20 0.34
CA2 P00918 1/20 0.34
PTGDR2 Q9Y5Y4 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7425296 0.84 KEAP1 (0.42) MAPTKEAP1NFE2L2FFAR4EGFR
SCHEMBL7428942 0.84 KEAP1 (0.40) MAPTKEAP1NFE2L2FFAR4EGFR
SCHEMBL8249919 0.82 MAPT (0.43) MAPTKEAP1NFE2L2FFAR4EGFR
SCHEMBL5870095 0.82 MAPT (0.43) MAPTKEAP1NFE2L2FFAR4EGFR
SCHEMBL7427491 0.80 ENPP2 (0.45) FFAR4PDCD1CD274MAPK1
SCHEMBL8258434 0.76 MAPT (0.39) MAPTKEAP1NFE2L2PKMPDCD1
SCHEMBL7422452 0.74 GRN (0.44) MAPK1
SCHEMBL5869605 0.74 KEAP1 (0.43) MAPTKEAP1NFE2L2FFAR4CPB1
SCHEMBL8248789 0.74 KEAP1 (0.43) MAPTKEAP1NFE2L2FFAR4CPB1
SCHEMBL5869800 0.73 MME (0.42) MAPTKEAP1NFE2L2PKMCD274

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002039997-A2 ACE-2 MODULATING COMPOUNDS AND USE THEREOF MILLENNIUM PHARMACEUTICALS, INC. (US) 2002-05-23 WO claimed
WO-2002039997-A2 ACE-2 MODULATING COMPOUNDS AND USE THEREOF MILLENNIUM PHARMACEUTICALS, INC. (US) 2002-05-23 WO disclosed