SCHEMBL7425296

SCHEMBL7425296

CC(C)CC(NCC(C(=O)O)c1ccc(OCc2csc3ccc(Cl)cc23)cc1)C(=O)O

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.42
NFE2L2 Q16236 1/20 0.42
FFAR4 Q5NUL3 1/20 0.39
MAPT P10636 2/20 0.38
CPB1 P15086 1/20 0.37
CYP2A6 P11509 2/20 0.35
EPHX1 P07099 1/20 0.35
CA2 P00918 1/20 0.35
ALDH1A1 P00352 1/20 0.35
FFAR1 O14842 1/20 0.35
NR4A2 P43354 1/20 0.34
FFAR2 O15552 1/20 0.34
EGFR P00533 1/20 0.34
ERBB2 P04626 1/20 0.34
EPHA2 P29317 1/20 0.34
KDR P35968 1/20 0.34
EPHB4 P54760 1/20 0.34
KLKB1 P03952 1/20 0.34
MAPK1 P28482 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7428942 0.91 KEAP1 (0.40) KEAP1NFE2L2FFAR4MAPTCPB1
SCHEMBL7425294 0.84 MAPT (0.41) KEAP1NFE2L2FFAR4MAPTCPB1
SCHEMBL8248789 0.82 KEAP1 (0.43) KEAP1NFE2L2FFAR4MAPTCPB1
SCHEMBL5869605 0.82 KEAP1 (0.43) KEAP1NFE2L2FFAR4MAPTCPB1
SCHEMBL7424624 0.79 GRN (0.44) MAPTALDH1A1FFAR1MAPK1
SCHEMBL5869794 0.77 MME (0.42) KEAP1NFE2L2MAPTMAPK1
SCHEMBL5869800 0.77 MME (0.42) KEAP1NFE2L2MAPTMAPK1
SCHEMBL5870047 0.77 MME (0.42) KEAP1NFE2L2MAPTMAPK1
SCHEMBL7425531 0.77 MME (0.42) KEAP1NFE2L2MAPTMAPK1
SCHEMBL7425285 0.74 KEAP1 (0.43) KEAP1NFE2L2FFAR4MAPTCPB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002039997-A2 ACE-2 MODULATING COMPOUNDS AND USE THEREOF MILLENNIUM PHARMACEUTICALS, INC. (US) 2002-05-23 WO claimed