SCHEMBL7425602

SCHEMBL7425602

CC(C)CC(NCC(C(=O)O)c1nc(-c2ccncc2)cs1)C(=O)O

nearest known ligand 0.41

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 14/20 0.41
ROCK2 O75116 13/20 0.41
PARP1 P09874 1/20 0.40
PRKACA P17612 1/20 0.38
FNTA P49354 1/20 0.38
FNTB P49356 1/20 0.38
PGGT1B P53609 1/20 0.38
CAPN1 P07384 2/20 0.38
MEN1 O00255 1/20 0.38
STAT3 P40763 1/20 0.38
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7426239 0.93 MEN1 (0.43) CAPN1MEN1STAT3KMT2A
SCHEMBL7424812 0.86 SMN1; SMN2 (0.34) FNTAFNTBPGGT1BCAPN1MEN1
SCHEMBL7426448 0.85 GRN (0.44) CAPN1MEN1KMT2A
SCHEMBL7425252 0.81 CTSK (0.54) FNTAFNTBPGGT1BMEN1KMT2A
SCHEMBL4714130 0.80 MEN1 (0.46) MEN1STAT3KMT2A
SCHEMBL7419514 0.79 FNTA (0.38) FNTAFNTBPGGT1B
SCHEMBL7427413 0.79 CTSS (0.48) ROCK1ROCK2PRKACAFNTAFNTB
SCHEMBL7420389 0.79 CTSS (0.48) ROCK1ROCK2PRKACAFNTAFNTB
SCHEMBL4714337 0.76 CTSK (0.58)
SCHEMBL5869695 0.75 ROCK1 (0.42) ROCK1ROCK2PARP1PRKACAFNTA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002039997-A2 ACE-2 MODULATING COMPOUNDS AND USE THEREOF MILLENNIUM PHARMACEUTICALS, INC. (US) 2002-05-23 WO claimed
WO-2002039997-A2 ACE-2 MODULATING COMPOUNDS AND USE THEREOF MILLENNIUM PHARMACEUTICALS, INC. (US) 2002-05-23 WO disclosed