SCHEMBL7424812

SCHEMBL7424812

Cc1cc(C)cc(-c2csc(C(CNC(CC(C)C)C(=O)O)C(=O)O)n2)c1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.34
MAPT P10636 2/20 0.34
KDM4E B2RXH2 1/20 0.34
HTT P42858 1/20 0.34
ALDH1A1 P00352 3/20 0.34
TAS1R3 Q7RTX0 1/20 0.34
TAS1R1 Q7RTX1 1/20 0.34
CYP2C19 P33261 1/20 0.34
MAPK1 P28482 1/20 0.34
KMT2A Q03164 3/20 0.34
MEN1 O00255 2/20 0.34
CYP2C9 P11712 1/20 0.34
FNTA P49354 1/20 0.34
FNTB P49356 1/20 0.34
PGGT1B P53609 1/20 0.34
CAPN1 P07384 3/20 0.33
NPC1 O15118 2/20 0.33
RAB9A P51151 2/20 0.33
STAT3 P40763 1/20 0.33
GFER P55789 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7426448 0.88 GRN (0.44) SMN1; SMN2MAPTKDM4EHTTALDH1A1
SCHEMBL7426239 0.88 MEN1 (0.43) SMN1; SMN2MAPTKDM4EHTTALDH1A1
SCHEMBL7425602 0.86 ROCK1 (0.41) KMT2AMEN1FNTAFNTBPGGT1B
SCHEMBL7423334 0.84 DHFR (0.34) MAPTALDH1A1TAS1R3TAS1R1CYP2C19
SCHEMBL7426736 0.81 CTSK (0.48) SMN1; SMN2MAPTKDM4EHTTALDH1A1
SCHEMBL7417292 0.78 ALDH1A1 (0.34) MAPTKDM4EALDH1A1TAS1R3TAS1R1
SCHEMBL5869832 0.76 ACE2 (0.38) SMN1; SMN2MAPTKDM4EHTTALDH1A1
SCHEMBL7426920 0.75 CTSK (0.38) MAPTKDM4EALDH1A1TAS1R3TAS1R1
SCHEMBL7417825 0.74 GRN (0.43) MAPTHTTALDH1A1MAPK1GRN
SCHEMBL7382345 0.74 CTSK (0.41) SMN1; SMN2MAPTHTTALDH1A1CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002039997-A2 ACE-2 MODULATING COMPOUNDS AND USE THEREOF MILLENNIUM PHARMACEUTICALS, INC. (US) 2002-05-23 WO claimed
WO-2002039997-A2 ACE-2 MODULATING COMPOUNDS AND USE THEREOF MILLENNIUM PHARMACEUTICALS, INC. (US) 2002-05-23 WO disclosed