SCHEMBL7425815

SCHEMBL7425815

CC(C)CC(NCC(C(=O)O)c1nc(Cc2cc(Cl)cc(Cl)c2)co1)C(=O)O

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GRN P28799 5/20 0.43
SORT1 Q99523 5/20 0.43
ACE2 Q9BYF1 4/20 0.40
ACE P12821 3/20 0.40
ALDH1A1 P00352 1/20 0.35
LMNA P02545 1/20 0.35
MAPK1 P28482 1/20 0.34
DHFR P00374 1/20 0.33
MAPT P10636 1/20 0.33
HTT P42858 1/20 0.33
TYR P14679 1/20 0.32
C3AR1 Q16581 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7425447 0.88 DHFR (0.34) GRNSORT1ALDH1A1MAPK1DHFR
SCHEMBL7425011 0.84 GRN (0.44) GRNSORT1ACE2ACEALDH1A1
SCHEMBL7421108 0.82 SORT1 (0.42) GRNSORT1ACE2ACEALDH1A1
SCHEMBL7417825 0.79 GRN (0.43) GRNSORT1ACE2ACEALDH1A1
SCHEMBL7424365 0.77 GRN (0.43) GRNSORT1ACE2ACEALDH1A1
SCHEMBL7419023 0.77 GRN (0.47) GRNSORT1ACE2ACEALDH1A1
SCHEMBL5869871 0.77 ACE2 (0.53) GRNSORT1ACE2ACEALDH1A1
SCHEMBL8249951 0.77 ACE2 (0.53) GRNSORT1ACE2ACEALDH1A1
SCHEMBL7423860 0.76 SORT1 (0.44) GRNSORT1ACE2ACEALDH1A1
SCHEMBL7419079 0.76 BCHE (0.37) ALDH1A1MAPK1C3AR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002039997-A2 ACE-2 MODULATING COMPOUNDS AND USE THEREOF MILLENNIUM PHARMACEUTICALS, INC. (US) 2002-05-23 WO claimed
WO-2002039997-A2 ACE-2 MODULATING COMPOUNDS AND USE THEREOF MILLENNIUM PHARMACEUTICALS, INC. (US) 2002-05-23 WO disclosed