SCHEMBL7425874

SCHEMBL7425874

Cc1cccc2[nH]c(C(=O)C(C)(C)[C@H](N)C(=O)NC(CC(=O)O)C(=O)COc3ccccc3C(N)=O)c(C)c12

nearest known ligand 0.46

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 7/20 0.46
CASP3 P42574 8/20 0.39
PARP1 P09874 1/20 0.37
CASP6 P55212 4/20 0.37
CASP8 Q14790 4/20 0.37
MAPT P10636 2/20 0.35
ALDH1A1 P00352 1/20 0.35
MEN1 O00255 1/20 0.33
POLB P06746 1/20 0.33
KMT2A Q03164 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7535926 0.83 CASP3 (0.48) CASP3CASP6CASP8
SCHEMBL5970178 0.83 CASP1 (0.32) CASP1
SCHEMBL5969967 0.83 CASP3 (0.39) CASP1CASP3CASP6CASP8
SCHEMBL5970067 0.83 PYGL (0.36) CASP1MAPTMEN1POLBKMT2A
SCHEMBL5970304 0.81 CASP1 (0.37) CASP1CASP3CASP6CASP8
SCHEMBL7536333 0.71 CASP3 (0.33) CASP1CASP3CASP6CASP8
SCHEMBL7540320 0.66 CASP3 (0.49) CASP3CASP6CASP8
SCHEMBL7537055 0.66
SCHEMBL7535127 0.62 CASP3 (0.47) CASP1CASP3CASP6CASP8
SCHEMBL6595219 0.62 MAP2 (0.42) PARP1MAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1159291-A1 C-TERMINAL MODIFIED (N-SUBSTITUTED)-2-INDOLYLCARBONYLDIPEPTIDES AS INHIBITORS OF THE ICE/CED-3 FAMILY OF CYSTEINE PROTEASES Idun Pharmaceuticals, Inc. (US) 2001-12-05 EP disclosed
WO-2001000658-A1 C-TERMINAL MODIFIED (N-SUBSTITUTED)-2-INDOLYLCARBONYLDIPEPTIDES AS INHIBITORS OF THE ICE/CED-3 FAMILY OF CYSTEINE PROTEASES IDUN PHARMACEUTICALS, INC. (US) 2001-01-04 WO disclosed