SCHEMBL7426014

SCHEMBL7426014

COc1ccc2[nH]c(C(=O)NC(CN[C@@H](CC(C)C)C(=O)O)C(=O)O)cc2c1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 9/20 0.61
MAPT P10636 6/20 0.61
ALDH1A1 P00352 6/20 0.61
PYGL P06737 1/20 0.57
TAS1R3 Q7RTX0 1/20 0.55
TAS1R1 Q7RTX1 1/20 0.55
CTSL P07711 1/20 0.53
CTSS P25774 1/20 0.53
NPC1 O15118 3/20 0.51
RAB9A P51151 3/20 0.51
PDGFRB P09619 1/20 0.50
PDGFRA P16234 1/20 0.50
LMNA P02545 1/20 0.50
HPGD P15428 1/20 0.50
HTT P42858 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
BCAT1 P54687 1/20 0.48
XDH P47989 1/20 0.47
HDAC6 Q9UBN7 2/20 0.47
MEN1 O00255 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5869272 0.84 KDM4E (0.58) KDM4EMAPTALDH1A1PYGLTAS1R3
SCHEMBL5869262 0.84 KDM4E (0.58) KDM4EMAPTALDH1A1PYGLTAS1R3
SCHEMBL5869279 0.84 KDM4E (0.58) KDM4EMAPTALDH1A1PYGLTAS1R3
SCHEMBL24019692 0.80 KDM4E (0.77) KDM4EMAPTALDH1A1PYGLNPC1
SCHEMBL5822796 0.78 TAS1R3 (0.58) KDM4EALDH1A1PYGLTAS1R3TAS1R1
SCHEMBL7426574 0.76 CTSL (0.59) ALDH1A1TAS1R3TAS1R1CTSLCTSS
SCHEMBL20853657 0.76 TAS1R3 (0.78) PYGLTAS1R3TAS1R1CTSLCTSS
SCHEMBL25517392 0.76 TAS1R3 (0.78) PYGLTAS1R3TAS1R1CTSLCTSS
SCHEMBL25197064 0.76 TAS1R3 (0.78) PYGLTAS1R3TAS1R1CTSLCTSS
SCHEMBL17149703 0.75 KDM4E (0.66) KDM4EMAPTALDH1A1PYGLNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002039997-A2 ACE-2 MODULATING COMPOUNDS AND USE THEREOF MILLENNIUM PHARMACEUTICALS, INC. (US) 2002-05-23 WO disclosed