SCHEMBL7426429

SCHEMBL7426429

NC(=O)c1cccc([C@H](Cc2ccccc2)C(=O)CNc2ccccc2)c1Oc1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SIRT2 Q8IXJ6 6/20 0.41
SIRT1 Q96EB6 2/20 0.41
FFAR1 O14842 7/20 0.39
CTNNB1 P35222 1/20 0.39
AURKA O14965 1/20 0.37
RPS6KB1 P23443 1/20 0.37
GNA15 P30679 1/20 0.36
PTGER3 P43115 1/20 0.36
FFAR4 Q5NUL3 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
PPARG P37231 3/20 0.36
PPARA Q07869 3/20 0.36
EPHX1 P07099 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7424973 0.86 MTNR1A (0.40) SIRT2SIRT1FFAR1CTNNB1AURKA
SCHEMBL5049439 0.65 CTNNB1 (0.59) SIRT2SIRT1CTNNB1
SCHEMBL8211650 0.65 CTNNB1 (0.54) SIRT2SIRT1CTNNB1AURKARPS6KB1
SCHEMBL27991301 0.64 CTNNB1 (0.57) SIRT2SIRT1CTNNB1TDP1
SCHEMBL27872615 0.64 CTNNB1 (0.57) SIRT2SIRT1CTNNB1
SCHEMBL27464948 0.64 CTNNB1 (0.53) SIRT2SIRT1CTNNB1
SCHEMBL20178657 0.63 EPHX1 (0.47) SIRT2EPHX1
SCHEMBL28081509 0.63 BCAT2 (0.61) SIRT2SIRT1CTNNB1AURKARPS6KB1
Diphenylether SCHEMBL23068684 0.62 CTNNB1 (0.74) SIRT2SIRT1CTNNB1
SCHEMBL9189752 0.62 CTNNB1 (0.62) SIRT2SIRT1CTNNB1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1073632-A1 SUBSTITUTED BENZAMIDES, THEIR PRODUCTION AND THEIR USE AS CYSTEINE PROTEASE INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 2001-02-07 EP disclosed
WO-1999054293-A1 SUBSTITUTED BENZAMIDES, THEIR PRODUCTION AND THEIR USE AS CYSTEINE PROTEASE INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 1999-10-28 WO disclosed