SCHEMBL7426447

SCHEMBL7426447

Nc1cc(-c2cccnc2)cc2nc(-c3ccccc3)nn12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 3/20 0.46
F12 P00748 1/20 0.45
SMN1; SMN2 Q16637 5/20 0.45
ALDH1A1 P00352 5/20 0.45
NPC1 O15118 2/20 0.45
HPGD P15428 2/20 0.45
RAB9A P51151 2/20 0.45
NFKB1 P19838 1/20 0.45
HTT P42858 1/20 0.45
NFKB2 Q00653 1/20 0.45
RELA Q04206 1/20 0.45
CYP2A6 P11509 2/20 0.44
CYP19A1 P11511 2/20 0.44
CYP17A1 P05093 1/20 0.44
CYP11B1 P15538 1/20 0.44
CYP11B2 P19099 1/20 0.44
ADORA1 P30542 2/20 0.43
ADORA2A P29274 1/20 0.43
POLB P06746 1/20 0.42
MEN1 O00255 3/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7423524 0.87 ALDH1A1 (0.53) ADORA3SMN1; SMN2ALDH1A1NPC1HPGD
SCHEMBL7428379 0.86 ADORA2A (0.53) F12SMN1; SMN2ALDH1A1NPC1HPGD
SCHEMBL7427474 0.86 SMN1; SMN2 (0.47) ADORA3SMN1; SMN2ALDH1A1NPC1HPGD
SCHEMBL7430129 0.84 CYP2A6 (0.51) ADORA3F12SMN1; SMN2ALDH1A1NPC1
SCHEMBL7426090 0.83 ADORA2A (0.56) ADORA2AMAPTF2HSD17B10
SCHEMBL7709122 0.81 MAOA (0.47) ADORA3SMN1; SMN2ALDH1A1NPC1HPGD
SCHEMBL7480172 0.79 RAB9A (0.46) SMN1; SMN2ALDH1A1NPC1HPGDRAB9A
SCHEMBL7703064 0.78 ALDH1A1 (0.45) ADORA3SMN1; SMN2ALDH1A1NPC1HPGD
SCHEMBL7542178 0.78 ADORA2A (0.52) ADORA3SMN1; SMN2ALDH1A1NPC1HPGD
SCHEMBL7151749 0.77 ALDH1A1 (0.49) ADORA3F12SMN1; SMN2ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1214322-A2 AMINO-TRIAZOLOPYRIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2002-06-19 EP disclosed
US-6355653-B1 DRUG AND CARRIER FOR ANTIALLERGENS, BRAIN DISORDERS AND NEUROTRANSMITTERS HOFFMANN-LA ROCHE INC. 2002-03-12 US disclosed
WO-2001017999-A2 AMINO-TRIAZOLOPYRIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2001-03-15 WO disclosed