SCHEMBL7426747

SCHEMBL7426747

CCOc1nc(C)c2cc(OC)c(OC)cc2c1C(=O)OC

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.42
KDM4E B2RXH2 3/20 0.42
GAA P10253 3/20 0.42
GABRA1 P14867 3/20 0.42
GABRA5 P31644 3/20 0.42
GABRA3 P34903 3/20 0.42
GABRA2 P47869 3/20 0.42
GABRA6 Q16445 3/20 0.42
DPP4 P27487 5/20 0.41
TNF P01375 1/20 0.40
MAPT P10636 2/20 0.39
GMNN O75496 1/20 0.39
LMNA P02545 1/20 0.39
CYP1A2 P05177 1/20 0.39
POLB P06746 1/20 0.39
CYP3A4 P08684 1/20 0.39
TSHR P16473 1/20 0.39
GABRG2 P18507 1/20 0.39
NFKB1 P19838 1/20 0.39
APEX1 P27695 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7447294 0.79 KDM4E (0.42) ALDH1A1KDM4EGAAGABRA1GABRA5
SCHEMBL10791069 0.69 KDM4E (0.56) ALDH1A1KDM4EGAADPP4MAPT
SCHEMBL7446369 0.69 MEN1 (0.40) ALDH1A1KDM4EGAADPP4TNF
SCHEMBL12325390 0.68 CYP3A4 (0.46) ALDH1A1KDM4EGAAMAPTLMNA
Hydrochloric Acid SCHEMBL27947697 0.68 KDM4E (0.46) ALDH1A1KDM4EGAAMAPTCYP1A2
SCHEMBL7428283 0.68 VCP (0.39) ALDH1A1KDM4EGAADPP4TNF
SCHEMBL7431845 0.67 HPGD (0.45) ALDH1A1KDM4EGAAGABRA1GABRA5
SCHEMBL13514137 0.67 PDE4D (0.42) ALDH1A1KDM4EGAAMAPTTSHR
SCHEMBL7426725 0.66 LMNA (0.43) ALDH1A1KDM4EGAAMAPTLMNA
SCHEMBL20562964 0.65 LMNA (0.43) ALDH1A1GAAMAPTLMNACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4880817-A O-functionalized derivatives of substituted isoquinolin-3-ols having cardiotonic and/or phosphodiesterase fraction III inhibiting properties and/or renal vasodilating properties ORTHO PHARMACEUTICAL CORPORATION (US) 1989-11-14 US disclosed