SCHEMBL7428283

SCHEMBL7428283

CCOc1cc2c(C)nc(OC(=O)CC)c([N+](=O)[O-])c2cc1OC

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
VCP P55072 1/20 0.39
NTSR1 P30989 1/20 0.39
DPP4 P27487 2/20 0.38
TNF P01375 3/20 0.37
ALDH1A1 P00352 2/20 0.36
KDM4E B2RXH2 2/20 0.36
GAA P10253 1/20 0.36
LMNA P02545 1/20 0.35
CASP3 P42574 1/20 0.35
SENP8 Q96LD8 1/20 0.35
SENP7 Q9BQF6 1/20 0.35
SENP6 Q9GZR1 1/20 0.35
MEN1 O00255 1/20 0.35
NPC1 O15118 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C19 P33261 1/20 0.35
RAB9A P51151 1/20 0.35
KMT2A Q03164 1/20 0.35
PDE3B Q13370 1/20 0.35
PDE3A Q14432 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7446369 0.90 MEN1 (0.40) NTSR1DPP4TNFALDH1A1KDM4E
SCHEMBL7440312 0.87 NCEH1 (0.40) NTSR1DPP4TNFALDH1A1KDM4E
SCHEMBL7437559 0.86 KMT2A (0.41) VCPTNFALDH1A1KDM4ELMNA
SCHEMBL7444368 0.85 NTSR1 (0.45) VCPNTSR1LMNACASP3SENP6
SCHEMBL7443770 0.84 KMT2A (0.47) NTSR1ALDH1A1KDM4EGAAMEN1
SCHEMBL9830708 0.82 MEN1 (0.44) NTSR1DPP4ALDH1A1KDM4EGAA
SCHEMBL7439631 0.81 MAPT (0.40) VCPALDH1A1KDM4EGAALMNA
SCHEMBL7444737 0.81 PDE3B (0.44) DPP4TNFALDH1A1GAALMNA
SCHEMBL7441183 0.80 LMNA (0.39) ALDH1A1KDM4ELMNACASP3SENP8
SCHEMBL7443752 0.72 KDM4E (0.36) ALDH1A1KDM4EMAPTBLMTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4880817-A O-functionalized derivatives of substituted isoquinolin-3-ols having cardiotonic and/or phosphodiesterase fraction III inhibiting properties and/or renal vasodilating properties ORTHO PHARMACEUTICAL CORPORATION (US) 1989-11-14 US claimed