SCHEMBL7428121

SCHEMBL7428121

O=C(CBr)CC(=O)c1ccncc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLOD2 O00469 3/20 0.60
CYP3A4 P08684 3/20 0.60
PLOD3 O60568 2/20 0.60
PLOD1 Q02809 2/20 0.60
CYP1A2 P05177 2/20 0.60
CYP2D6 P10635 2/20 0.60
CYP2C19 P33261 2/20 0.60
ALDH1A1 P00352 2/20 0.60
HPGD P15428 2/20 0.60
CYP2C9 P11712 1/20 0.60
HIF1A Q16665 1/20 0.60
KDM4E B2RXH2 3/20 0.48
MPO P05164 1/20 0.48
ADORA3 P0DMS8 1/20 0.48
CYP2A6 P11509 1/20 0.48
NAPRT Q6XQN6 1/20 0.45
LMNA P02545 2/20 0.44
GAA P10253 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
PTPN1 P18031 3/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL84572 0.83 GSK3B (0.60) PLOD2CYP3A4PLOD3PLOD1CYP1A2
SCHEMBL10948430 0.83 PLOD2 (0.83) PLOD2CYP3A4PLOD3PLOD1CYP1A2
Bromide SCHEMBL6118414 0.81 GSK3B (0.58) PLOD2CYP3A4PLOD3PLOD1CYP1A2
Bromide SCHEMBL66813 0.81 GSK3B (0.58) PLOD2CYP3A4PLOD3PLOD1CYP1A2
Hydrochloric Acid SCHEMBL899290 0.81 GSK3B (0.58) PLOD2CYP3A4PLOD3PLOD1CYP1A2
Bromide SCHEMBL2773952 0.79 GSK3B (0.56) PLOD2CYP3A4PLOD3PLOD1CYP1A2
SCHEMBL1038505 0.79 PTPN1 (0.68) PLOD2CYP3A4PLOD3PLOD1CYP1A2
SCHEMBL200805 0.77 PLOD2 (0.73) PLOD2CYP3A4PLOD3PLOD1CYP1A2
SCHEMBL11599481 0.76 GSK3B (0.70) ALDH1A1HPGDKDM4ELMNAGAA
SCHEMBL27908337 0.76 ALDH1A1 (0.55) PLOD2CYP3A4PLOD3PLOD1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0329070-A1 Cardiotonic alkanoyl and aroyl oxazolones MERRELL DOW PHARMACEUTICALS INC. (US) 1989-08-23 EP disclosed