SCHEMBL7428133

SCHEMBL7428133

CC(C)CC(NCC(C(=O)O)c1coc(-c2ccccc2)n1)C(=O)O

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 2/20 0.40
HDAC8 Q9BY41 2/20 0.40
HDAC6 Q9UBN7 2/20 0.40
ALDH1A1 P00352 1/20 0.39
GRN P28799 1/20 0.39
SORT1 Q99523 1/20 0.39
CTSK P43235 1/20 0.38
PPARG P37231 3/20 0.38
PPARA Q07869 3/20 0.38
MMP1 P03956 1/20 0.38
MMP3 P08254 1/20 0.38
NPC1 O15118 1/20 0.38
POLB P06746 1/20 0.38
RAB9A P51151 1/20 0.38
MME P08473 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7423860 0.87 SORT1 (0.44) ALDH1A1GRNSORT1
SCHEMBL7417318 0.79 CNR2 (0.40) ALDH1A1GRNSORT1MME
SCHEMBL1655302 0.78 CTSK (0.62) HDAC1HDAC8HDAC6GRNSORT1
SCHEMBL5869312 0.77 ALDH1A1 (0.42) ALDH1A1PPARGPPARANPC1POLB
SCHEMBL6930381 0.77 ALDH1A1 (0.42) ALDH1A1PPARGPPARANPC1POLB
SCHEMBL7377704 0.77 GRN (0.43) ALDH1A1GRNSORT1CTSKMME
SCHEMBL7378949 0.76 MME (0.50) ALDH1A1CTSKMME
SCHEMBL7429293 0.75 SORT1 (0.34) ALDH1A1GRNSORT1POLB
SCHEMBL7421108 0.74 SORT1 (0.42) ALDH1A1GRNSORT1
SCHEMBL5869970 0.74 PPARG (0.46) HDAC1HDAC8HDAC6ALDH1A1PPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002039997-A2 ACE-2 MODULATING COMPOUNDS AND USE THEREOF MILLENNIUM PHARMACEUTICALS, INC. (US) 2002-05-23 WO claimed
WO-2002039997-A2 ACE-2 MODULATING COMPOUNDS AND USE THEREOF MILLENNIUM PHARMACEUTICALS, INC. (US) 2002-05-23 WO disclosed