SCHEMBL7429293

SCHEMBL7429293

Cc1cc(C)cc(Cc2nc(C(CNC(CC(C)C)C(=O)O)C(=O)O)co2)c1

nearest known ligand 0.34

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SORT1 Q99523 3/20 0.34
ALDH1A1 P00352 3/20 0.34
DHFR P00374 1/20 0.33
MMP2 P08253 1/20 0.33
CYP2C19 P33261 1/20 0.33
MAPK1 P28482 1/20 0.33
TAS1R3 Q7RTX0 1/20 0.33
TAS1R1 Q7RTX1 1/20 0.33
KMT2A Q03164 3/20 0.32
POLB P06746 2/20 0.32
ITGAV P06756 1/20 0.32
TYR P14679 1/20 0.32
GRN P28799 2/20 0.31
KLKB1 P03952 1/20 0.31
PYGL P06737 1/20 0.31
MEN1 O00255 1/20 0.31
CYP2C9 P11712 1/20 0.31
ELANE P08246 1/20 0.31
KDM4E B2RXH2 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7421108 0.89 SORT1 (0.42) SORT1ALDH1A1DHFRMAPK1GRN
SCHEMBL7425447 0.82 DHFR (0.34) SORT1ALDH1A1DHFRMMP2CYP2C19
SCHEMBL7426920 0.80 CTSK (0.38) SORT1ALDH1A1DHFRMMP2CYP2C19
SCHEMBL5869629 0.77 ACE2 (0.39) SORT1ALDH1A1MMP2CYP2C19MAPK1
SCHEMBL7423334 0.76 DHFR (0.34) SORT1ALDH1A1DHFRMMP2CYP2C19
SCHEMBL7421752 0.76 MEN1 (0.39) ALDH1A1CYP2C19KMT2AMEN1
SCHEMBL7428133 0.75 HDAC1 (0.40) SORT1ALDH1A1POLBGRN
SCHEMBL7417292 0.74 ALDH1A1 (0.34) SORT1ALDH1A1CYP2C19MAPK1TAS1R3
SCHEMBL7423860 0.74 SORT1 (0.44) SORT1ALDH1A1MAPK1GRN
SCHEMBL7426736 0.73 CTSK (0.48) SORT1ALDH1A1CYP2C19MAPK1TAS1R3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002039997-A2 ACE-2 MODULATING COMPOUNDS AND USE THEREOF MILLENNIUM PHARMACEUTICALS, INC. (US) 2002-05-23 WO claimed
WO-2002039997-A2 ACE-2 MODULATING COMPOUNDS AND USE THEREOF MILLENNIUM PHARMACEUTICALS, INC. (US) 2002-05-23 WO disclosed