SCHEMBL7428434

SCHEMBL7428434

CCC[CH]C(=O)NC1CCCN(S(=O)(=O)c2cccs2)CC1=O

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.48
KMT2A Q03164 3/20 0.48
KDM4E B2RXH2 1/20 0.46
MAPT P10636 1/20 0.45
RAB9A P51151 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
EPHX2 P34913 2/20 0.44
HTT P42858 1/20 0.44
ALDH1A1 P00352 2/20 0.44
GAA P10253 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
POLB P06746 1/20 0.43
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
PKM P14618 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7427117 0.88 MEN1 (0.52) MEN1KMT2AKDM4EMAPTRAB9A
SCHEMBL7042609 0.85 MEN1 (0.48) MEN1KMT2AKDM4EMAPTRAB9A
SCHEMBL7428439 0.84 MEN1 (0.48) MEN1KMT2AKDM4EMAPTRAB9A
SCHEMBL7481625 0.82 CTSK (0.39) SMN1; SMN2HTTALDH1A1GAA
SCHEMBL7426096 0.80 CTSK (0.54)
SCHEMBL7538673 0.80 ATM (0.49) KDM4EMAPTSMN1; SMN2HTTALDH1A1
SCHEMBL7427121 0.79 MEN1 (0.55) MEN1KMT2AKDM4EMAPTRAB9A
SCHEMBL6897906 0.79 CTSK (0.53) MEN1KMT2APKM
SCHEMBL7533624 0.79 CTSK (0.42) RAB9ASMN1; SMN2ALDH1A1GAACYP1A2
SCHEMBL7042614 0.78 MEN1 (0.51) MEN1KMT2AKDM4EMAPTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1158986-A4 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORP (US) 2002-03-27 EP claimed
EP-1158986-A1 PROTEASE INHIBITORS SmithKline Beecham Corporation (US) 2001-12-05 EP claimed
WO-2000038687-A1 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2000-07-06 WO claimed