SCHEMBL7533624

SCHEMBL7533624

CCC[CH]C(=O)NC1CCCN(S(=O)(=O)c2ncccc2C)CC1=O

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CTSK P43235 9/20 0.42
CTSL P07711 7/20 0.42
CTSS P25774 7/20 0.42
CTSB P07858 5/20 0.40
CTSV O60911 1/20 0.40
GAA P10253 1/20 0.38
ALDH1A1 P00352 1/20 0.37
TP53 P04637 2/20 0.36
LMNA P02545 1/20 0.36
CYP1A2 P05177 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
RAB9A P51151 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5096354 0.85 CTSK (0.43) CTSKCTSLCTSSCTSBCTSV
SCHEMBL7426096 0.85 CTSK (0.54) CTSKCTSLCTSSCTSBCTSV
SCHEMBL7533634 0.85 CTSK (0.42) CTSKCTSLCTSSCTSBCTSV
SCHEMBL7538673 0.83 ATM (0.49) GAAALDH1A1LMNASMN1; SMN2
SCHEMBL7481625 0.80 CTSK (0.39) CTSKCTSLCTSSCTSBCTSV
SCHEMBL5096358 0.79 CTSK (0.53) CTSKCTSLCTSSCTSBCTSV
SCHEMBL7428434 0.79 MEN1 (0.48) GAAALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL6897906 0.77 CTSK (0.53) CTSKCTSLCTSSCTSBCTSV
SCHEMBL7424838 0.76 CTSK (0.34) CTSKCTSLCTSSCTSBCTSV
SCHEMBL5093270 0.75 CTSK (0.52) CTSKCTSLCTSSCTSBCTSV

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1158986-A4 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORP (US) 2002-03-27 EP claimed
EP-1158986-A1 PROTEASE INHIBITORS SmithKline Beecham Corporation (US) 2001-12-05 EP claimed
WO-2000038687-A1 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2000-07-06 WO claimed