SCHEMBL7428707

SCHEMBL7428707

CCc1ccc[c]c1C(=N)N

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 2/20 0.38
GABRB2 P47870 2/20 0.38
GRIN2D O15399 1/20 0.35
GRIN3B O60391 1/20 0.35
GRIN1 Q05586 1/20 0.35
GRIN2A Q12879 1/20 0.35
GRIN2B Q13224 1/20 0.35
GRIN2C Q14957 1/20 0.35
GRIN3A Q8TCU5 1/20 0.35
SIGMAR1 Q99720 1/20 0.35
PRSS1 P07477 2/20 0.32
PRSS2 P07478 2/20 0.32
PRSS3 P35030 2/20 0.32
F2 P00734 2/20 0.32
TMPRSS6 Q8IU80 1/20 0.32
ST14 Q9Y5Y6 1/20 0.32
IDO1 P14902 2/20 0.32
CACNA1C Q13936 1/20 0.31
SCN5A Q14524 1/20 0.31
ALDH1A1 P00352 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6967624 0.81 SIGMAR1 (0.38) GABRA1GABRB2GRIN2DGRIN3BGRIN1
SCHEMBL5932184 0.77 GABRA1 (0.40) GABRA1GABRB2ALDH1A1GAAMAPT
SCHEMBL6633093 0.75 PRSS1 (0.36) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL14721446 0.73 ALDH1A1 (0.39) GABRA1GABRB2ALDH1A1GAAMAPT
SCHEMBL5907451 0.72 F2 (0.34) PRSS1PRSS2PRSS3F2F10
SCHEMBL6987504 0.72 F2 (0.34) PRSS1PRSS2PRSS3F2ALDH1A1
SCHEMBL17559557 0.71 ALDH1A1 (0.43) ALDH1A1
SCHEMBL18301295 0.70 CA1 (0.43) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL9853537 0.70 ALDH1A1 (0.41) GABRA1GABRB2GRIN2DGRIN3BGRIN1
SCHEMBL1933231 0.70

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1206444-A1 COMPOUNDS THAT INHIBIT TRYPTASE ACTIVITY Morphochem AG (DE) 2002-05-22 EP disclosed
WO-2001014320-A1 COMPOUNDS THAT INHIBIT TRYPTASE ACTIVITY MORPHOCHEM AG (DE) 2001-03-01 WO disclosed