SCHEMBL7429016

SCHEMBL7429016

CC(C)(C)OC(=O)NCc1ccc(N(CC(=O)O)C(=O)c2ccccc2)cc1CNC(=O)OC(C)(C)C.NC(=O)c1ccc2c(c1)CCC2

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
HDAC1 Q13547 2/20 0.34
MAPK14 Q16539 2/20 0.34
AVPR2 P30518 2/20 0.33
HDAC10 Q969S8 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
OPRM1 P35372 3/20 0.33
OPRD1 P41143 3/20 0.33
OPRK1 P41145 3/20 0.33
NR1H4 Q96RI1 1/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
MEN1 O00255 1/20 0.32
MAPT P10636 1/20 0.32
KMT2A Q03164 1/20 0.32
KDM4E B2RXH2 1/20 0.32
KDM4A O75164 1/20 0.32
RXRA P19793 1/20 0.32
RXRB P28702 1/20 0.32
RXRG P48443 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7430527 0.94 PDK1 (0.34) NPC1RAB9AHDAC1MAPK14AVPR2
SCHEMBL7430920 0.93 PDK1 (0.34) NPC1RAB9AHDAC1MAPK14AVPR2
SCHEMBL5210913 0.85 NPC1 (0.39) NPC1RAB9AHDAC1MAPK14NR1H4
SCHEMBL5210889 0.85 NPC1 (0.40) NPC1RAB9AHDAC1MAPK14OPRM1
SCHEMBL5210074 0.84 RXRB (0.38) NPC1RAB9AHDAC1MAPK14NR1H4
Trifluoroacetic Acid SCHEMBL4807978 0.84 NPC1 (0.37) NPC1RAB9AHDAC1MAPK14SMN1; SMN2
SCHEMBL5216930 0.83 RAB9A (0.37) NPC1RAB9AHDAC1MAPK14SMN1; SMN2
SCHEMBL7131862 0.80 RXRA (0.36) NPC1RAB9AMAPK14OPRM1OPRD1
Hydrochloric Acid SCHEMBL7427799 0.80 MAPK14 (0.36) NPC1RAB9AMAPK14OPRM1OPRD1
Hydrochloric Acid SCHEMBL7128388 0.80 RXRA (0.36) NPC1RAB9AMAPK14OPRM1OPRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1192135-A2 SERINE PROTEASE INHIBITORS ELI LILLY AND COMPANY (US) 2002-04-03 EP disclosed
WO-2000076970-A2 SERINE PROTEASE INHIBITORS ELI LILLY AND COMPANY (US) 2000-12-21 WO disclosed