SCHEMBL7430920

SCHEMBL7430920

CC(C)(C)OC(=O)NCc1cc(N(CC(=O)O)C(=O)c2ccccc2)ccc1C(=O)O.NC(=O)c1ccc2c(c1)CCC2

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDK1 Q15118 1/20 0.34
PDK2 Q15119 1/20 0.34
PDK3 Q15120 1/20 0.34
PDK4 Q16654 1/20 0.34
ALDH1A1 P00352 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
HDAC1 Q13547 1/20 0.33
MAPK14 Q16539 2/20 0.33
RXRA P19793 1/20 0.33
RXRB P28702 1/20 0.33
RXRG P48443 1/20 0.33
AVPR2 P30518 2/20 0.32
METAP2 P50579 1/20 0.32
HDAC10 Q969S8 1/20 0.32
HDAC6 Q9UBN7 1/20 0.32
PPARG P37231 1/20 0.32
PPARA Q07869 1/20 0.32
OPRM1 P35372 1/20 0.32
OPRD1 P41143 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7430527 0.96 PDK1 (0.34) PDK1PDK2PDK3PDK4NPC1
SCHEMBL7429016 0.93 NPC1 (0.35) PDK1PDK2PDK3PDK4NPC1
SCHEMBL5210074 0.84 RXRB (0.38) PDK1PDK2PDK3PDK4ALDH1A1
SCHEMBL5210913 0.83 NPC1 (0.39) NPC1RAB9AHDAC1MAPK14RXRA
SCHEMBL5210889 0.83 NPC1 (0.40) NPC1RAB9AHDAC1MAPK14RXRA
Trifluoroacetic Acid SCHEMBL4807978 0.82 NPC1 (0.37) NPC1RAB9AHDAC1MAPK14RXRA
SCHEMBL5216930 0.81 RAB9A (0.37) ALDH1A1NPC1RAB9AHDAC1MAPK14
Trifluoroacetic Acid SCHEMBL7433400 0.81 ALDH1A1 (0.37) ALDH1A1NPC1RAB9AMAPK14RXRA
SCHEMBL7131862 0.80 RXRA (0.36) ALDH1A1NPC1RAB9AMAPK14RXRA
Hydrochloric Acid SCHEMBL7128388 0.79 RXRA (0.36) ALDH1A1NPC1RAB9AMAPK14RXRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1240154-A1 SERINE PROTEASE INHIBITORS Tularik Limited (GB) 2002-09-18 EP disclosed
WO-2001044226-A1 SERINE PROTEASE INHIBITORS TULARIK LIMITED (GB) 2001-06-21 WO disclosed