Bicarbonate

Bicarbonate

SCHEMBL7429705

Cc1cc(C(=O)NCc2ccc(F)cc2)c(NC(=O)C2CCCCC2)s1.O=C(O)O

nearest known ligand 0.45

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

GSK3AGSK3BIMPA1

The experimentally established mechanism targets of Bicarbonate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.45
POLB P06746 2/20 0.43
RAB9A P51151 1/20 0.43
HDAC6 Q9UBN7 1/20 0.42
ALDH1A1 P00352 3/20 0.42
CYP2C19 P33261 2/20 0.42
MAPT P10636 2/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP1A2 P05177 1/20 0.42
KMT2A Q03164 1/20 0.42
KDM4E B2RXH2 1/20 0.42
LMNA P02545 1/20 0.42
REV1 Q9UBZ9 1/20 0.41
CNR2 P34972 1/20 0.41
SMO Q99835 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7429703 0.91 MMP13 (0.43) SMN1; SMN2ALDH1A1CYP2C19MAPTCYP1A2
Bicarbonate SCHEMBL7890842 0.91 ALDH1A1 (0.50) SMN1; SMN2RAB9AHDAC6ALDH1A1CYP2C19
Bicarbonate SCHEMBL7420725 0.88 POLB (0.49) SMN1; SMN2POLBRAB9AHDAC6ALDH1A1
Bicarbonate SCHEMBL7427368 0.88 SMN1; SMN2 (0.45) SMN1; SMN2POLBRAB9AHDAC6ALDH1A1
SCHEMBL8250085 0.87 REV1 (0.45) SMN1; SMN2POLBALDH1A1CYP2C19MAPT
Bicarbonate SCHEMBL7886928 0.85 POLB (0.48) SMN1; SMN2POLBRAB9AALDH1A1KMT2A
Bicarbonate SCHEMBL7881463 0.84 ALDH1A1 (0.53) SMN1; SMN2POLBRAB9AALDH1A1MAPT
Bicarbonate SCHEMBL7421198 0.82 TSHR (0.44) RAB9AKMT2ALMNAREV1
SCHEMBL7890839 0.81 ALDH1A1 (0.45) POLBALDH1A1CYP2C19MAPTCYP3A4
Bicarbonate SCHEMBL7890931 0.81 SMN1; SMN2 (0.51) SMN1; SMN2POLBRAB9AALDH1A1CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0934301-A1 AMINOTHIOPHENE CARBOXYLIC ACID AMIDES AND THE USE THEREOF AS PHOSPHODIESTERASE INHIBITORS MERCK PATENT GmbH (DE) 1999-08-11 EP disclosed
WO-1998016521-A1 AMINOTHIOPHENE CARBOXYLIC ACID AMIDES AND THE USE THEREOF AS PHOSPHODIESTERASE INHIBITORS MERCK PATENT GMBH (DE) 1998-04-23 WO disclosed