SCHEMBL7430478

SCHEMBL7430478

COc1cc2c(c([N+](=O)[O-])c1O)C(=O)c1ccccc1C2=O

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.54
RAB9A P51151 4/20 0.54
MAPT P10636 4/20 0.54
MEN1 O00255 3/20 0.54
KMT2A Q03164 3/20 0.54
ALDH1A1 P00352 3/20 0.52
CYP3A4 P08684 1/20 0.52
TSHR P16473 1/20 0.52
MAOA P21397 2/20 0.48
SMN1; SMN2 Q16637 3/20 0.48
KDM4E B2RXH2 1/20 0.47
USP2 O75604 1/20 0.47
DUSP3 P51452 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
PGAM1 P18669 4/20 0.47
HPGD P15428 1/20 0.45
BCL2 P10415 1/20 0.44
MCL1 Q07820 1/20 0.44
LCK P06239 1/20 0.44
GLA P06280 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11577441 0.81 ALDH1A1 (0.68) NPC1RAB9AMAPTMEN1KMT2A
SCHEMBL7435273 0.81 BCL2 (0.63) NPC1RAB9AMAPTMEN1KMT2A
SCHEMBL23199010 0.81 MAPT (0.69) NPC1RAB9AMAPTMEN1KMT2A
SCHEMBL14379281 0.80 MAPT (0.51) NPC1RAB9AMAPTMEN1KMT2A
SCHEMBL18601894 0.79 RAB9A (0.62) NPC1RAB9AMAPTMEN1KMT2A
SCHEMBL1609981 0.78 GAA (0.41) MAPTMEN1KMT2AALDH1A1KDM4E
SCHEMBL11515026 0.77 ALDH1A1 (0.56) NPC1RAB9AMAPTMEN1KMT2A
SCHEMBL16227229 0.76 MAPT (0.65) NPC1RAB9AMAPTMEN1KMT2A
SCHEMBL31237408 0.76 MAPT (0.65) NPC1RAB9AMAPTMEN1KMT2A
SCHEMBL23198991 0.76 EPHX2 (0.65) NPC1RAB9AMAPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20020037931-A1 Substituted nitrated catechols, their use in the treatment of some central and peripheral nervous system disorders and pharmaceutical compositions containing them PORTELA & C.A., S.A. (PT) 2002-03-28 US disclosed
EP-1167341-A1 Substituted nitrated catechols, their use in the treatment of some central and peripheral nervous system disorders and pharmaceutical compositions containing them Portela & Ca., S.A. (PT) 2002-01-02 EP disclosed
WO-2001098250-A1 SUBSTITUTED NITRATED CATECHOLS, THEIR USE IN THE TREATMENT OF SOME CENTRAL AND PERIPHERAL NERVOUS SYSTEM DISORDERS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM PORTELA & CA SA (PT) 2001-12-27 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020037931-A1 Substituted nitrated catechols, their use in the treatment of some central and peripheral nervous system disorders and pharmaceutical compositions containing them SLC6A2, COMT, SLC6A3 NPC1 930/4885RAB9A 3311/4885MAPT 379/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.