SCHEMBL7430843

SCHEMBL7430843

O=C1NC(=O)c2c1c(OP(=O)(O)O)cc1ccccc21

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR84 Q9NQS5 4/20 0.41
INPPL1 O15357 7/20 0.39
INPP5A Q14642 4/20 0.39
INPP5B P32019 2/20 0.39
SRC P12931 3/20 0.37
ALDH1A1 P00352 2/20 0.37
KDM4E B2RXH2 1/20 0.37
USP2 O75604 1/20 0.37
HPGD P15428 1/20 0.37
PDE3A Q14432 1/20 0.37
HSD17B10 Q99714 1/20 0.37
MAPT P10636 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
AKT1 P31749 1/20 0.36
CDK4 P11802 2/20 0.35
CCND1 P24385 2/20 0.35
GSK3A P49840 2/20 0.35
GSK3B P49841 2/20 0.35
CDK5 Q00535 2/20 0.35
CDK5R1 Q15078 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28295682 0.76 GPR84 (0.67) GPR84INPPL1INPP5AINPP5BSRC
SCHEMBL1029435 0.73 ALDH1A1 (0.42) ALDH1A1KDM4EMAPTNPSR1CDK4
SCHEMBL8094182 0.73 GSK3B (0.36) GPR84ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL8080577 0.73 CDK4 (0.36) GPR84ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL1756365 0.73 TRPM4 (0.48) MAPTCDK4CCND1GSK3AGSK3B
SCHEMBL297203 0.73 MAPT (0.53) GPR84INPPL1INPP5AINPP5BSRC
SCHEMBL789452 0.71 TRPM4 (0.47) MAPTCDK4CCND1GSK3AGSK3B
SCHEMBL1516404 0.70 ADORA2A (0.35) ALDH1A1MAPTNPSR1CDK4CCND1
SCHEMBL9438223 0.70 NQO2 (0.48) GPR84INPPL1INPP5AINPP5BSRC
SCHEMBL6848266 0.69 CDK4 (0.42) GPR84ALDH1A1KDM4EMAPTCDK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002047679-A2 NONPEPTIDE AGONISTS AND ANTAGONISTS OF VASOPRESSIN RECEPTORS EMORY UNIVERSITY (US) 2002-06-20 WO disclosed