SCHEMBL8094182

SCHEMBL8094182

O=C(CBr)Oc1cc2ccccc2c2c1C(=O)NC2=O

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 5/20 0.36
CDK4 P11802 3/20 0.36
CCND1 P24385 3/20 0.36
PTPN1 P18031 2/20 0.35
ALDH1A1 P00352 3/20 0.34
NPSR1 Q6W5P4 2/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
MAPT P10636 1/20 0.34
KDM4E B2RXH2 2/20 0.33
HPGD P15428 2/20 0.33
GPR84 Q9NQS5 1/20 0.33
GAA P10253 1/20 0.33
RXFP1 Q9HBX9 1/20 0.33
GSK3A P49840 2/20 0.33
CDK5 Q00535 2/20 0.33
CDK5R1 Q15078 2/20 0.33
KMT2A Q03164 2/20 0.32
LMNA P02545 1/20 0.32
POLB P06746 1/20 0.32
PTGS2 P35354 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8080577 0.86 CDK4 (0.36) GSK3BCDK4CCND1ALDH1A1NPSR1
SCHEMBL7430843 0.73 GPR84 (0.41) GSK3BCDK4CCND1ALDH1A1NPSR1
SCHEMBL8853276 0.72 CDK4 (0.40) GSK3BCDK4CCND1ALDH1A1NPSR1
SCHEMBL11466604 0.71 ALDH1A1 (0.56) PTPN1ALDH1A1L3MBTL1KDM4EHPGD
SCHEMBL28324766 0.71 ALDH1A1 (0.44) PTPN1ALDH1A1L3MBTL1MAPTKDM4E
SCHEMBL1029435 0.70 ALDH1A1 (0.42) GSK3BCDK4CCND1ALDH1A1NPSR1
SCHEMBL3852137 0.70 CDK4 (0.44) GSK3BCDK4CCND1ALDH1A1NPSR1
SCHEMBL1756365 0.70 TRPM4 (0.48) GSK3BCDK4CCND1MAPTGSK3A
SCHEMBL9556428 0.69 CDK4 (0.39) GSK3BCDK4CCND1MAPTGPR84
SCHEMBL789452 0.68 TRPM4 (0.47) GSK3BCDK4CCND1MAPTGSK3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6160128-A Tritioacetylating reagents and processes for preparation thereof THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2000-12-12 US disclosed