SCHEMBL7432011

SCHEMBL7432011

CC(=O)SCC(Cc1ccc(F)cc1)C(=O)Nc1cccc(C(=O)O)c1.[NaH]

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.45
PPARA Q07869 6/20 0.44
MME P08473 1/20 0.44
ACE P12821 1/20 0.44
KMT2A Q03164 4/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
ABCC3 O15438 1/20 0.43
NR1I2 O75469 1/20 0.43
ABCB11 O95342 1/20 0.43
NR3C1 P04150 1/20 0.43
RARG P13631 1/20 0.43
CNR1 P21554 1/20 0.43
OPRK1 P41145 1/20 0.43
NR1H2 P55055 1/20 0.43
NR1H3 Q13133 1/20 0.43
NR1I3 Q14994 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7432902 0.99 ALDH1A1 (0.46) ALDH1A1PPARAMMEACEKMT2A
SCHEMBL392082 0.90 ALDH1A1 (0.52) ALDH1A1PPARAMMEACEKMT2A
SCHEMBL7431904 0.89 NR1H4 (0.48) ALDH1A1PPARAMMEACEKMT2A
SCHEMBL7432008 0.89 KMT2A (0.43) ALDH1A1PPARAMMEACEKMT2A
SCHEMBL7429797 0.88 PPARA (0.48) ALDH1A1PPARAKMT2ACYP1A2CYP3A4
SCHEMBL7431217 0.88 KCNK3 (0.46) ALDH1A1PPARAMMEACEKMT2A
SCHEMBL7431596 0.87 NPC1 (0.49) ALDH1A1PPARAKMT2ACYP1A2CYP3A4
SCHEMBL7435916 0.86 PPARA (0.45) ALDH1A1PPARAMMEACEKMT2A
SCHEMBL7435223 0.82 FOLH1 (0.52) ALDH1A1PPARAPTGER4
SCHEMBL7397309 0.82 PARP1 (0.50) ALDH1A1PPARAMMEACEKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5210266-A Analgesic enkephalinase inhibitors DAINIPPON PHARMACEUTICAL CO., LTD. (JP) 1993-05-11 US disclosed
US-5179125-A Analgesics DAINIPPON PHARMACEUTICAL CO., LTD. (JP) 1993-01-12 US disclosed
EP-0318859-A2 N-substituted mercaptopropanamide derivatives Dainippon Pharmaceutical Co., Ltd. (JP) 1989-06-07 EP disclosed