SCHEMBL7433225

SCHEMBL7433225

CC(C)(C)C(=O)OCOC(=O)c1cccc(N)c1

nearest known ligand 0.54

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 2/20 0.54
ADRB1 P08588 2/20 0.54
ADRB3 P13945 2/20 0.54
CHRNB2 P17787 1/20 0.47
CHRNA4 P43681 1/20 0.47
PBRM1 Q86U86 1/20 0.42
ALDH1A1 P00352 2/20 0.42
ELANE P08246 3/20 0.42
LMNA P02545 2/20 0.41
NPC1 O15118 1/20 0.41
MITF O75030 1/20 0.41
POLB P06746 1/20 0.41
KDM4E B2RXH2 1/20 0.40
HTR7 P34969 1/20 0.39
RXRA P19793 1/20 0.39
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
MAOA P21397 1/20 0.38
LOXL2 Q9Y4K0 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19354448 0.84 ADRB2 (0.53) ADRB2ADRB1ADRB3NPC1KDM4E
SCHEMBL14034889 0.81 LMNA (0.59) ADRB2ADRB1ADRB3ALDH1A1LMNA
SCHEMBL18862636 0.81 MAPK1 (0.55) ADRB2ADRB1ADRB3ALDH1A1ELANE
SCHEMBL8123928 0.79 KDM4E (0.40) ADRB2ADRB1ADRB3ALDH1A1ELANE
SCHEMBL29465556 0.78 LMNA (0.62) ADRB2ADRB1ADRB3CHRNB2CHRNA4
SCHEMBL133366 0.78 LMNA (0.62) ADRB2ADRB1ADRB3CHRNB2CHRNA4
SCHEMBL1802562 0.77 ADRB2 (0.55) ADRB2ADRB1ADRB3CHRNB2CHRNA4
Hydrochloric Acid SCHEMBL642777 0.76 LMNA (0.61) ADRB2ADRB1ADRB3CHRNB2CHRNA4
Methane SCHEMBL15286491 0.76 LMNA (0.61) ADRB2ADRB1ADRB3CHRNB2CHRNA4
SCHEMBL1509380 0.76 MAPK1 (0.62) ADRB2ADRB1ADRB3CHRNB2CHRNA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5210266-A Analgesic enkephalinase inhibitors DAINIPPON PHARMACEUTICAL CO., LTD. (JP) 1993-05-11 US disclosed
US-5179125-A Analgesics DAINIPPON PHARMACEUTICAL CO., LTD. (JP) 1993-01-12 US disclosed
EP-0318859-A2 N-substituted mercaptopropanamide derivatives Dainippon Pharmaceutical Co., Ltd. (JP) 1989-06-07 EP disclosed