SCHEMBL7433585

SCHEMBL7433585

CCCCC(NCC(CC(C)C)NC(=O)c1coc2ccccc12)C(=O)CSCc1ccco1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 2/20 0.35
ALDH1A1 P00352 6/20 0.35
POLB P06746 4/20 0.35
USP2 O75604 2/20 0.35
MAPT P10636 2/20 0.35
HSD17B10 Q99714 1/20 0.35
SMN1; SMN2 Q16637 2/20 0.33
HPGD P15428 2/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
CTSL P07711 2/20 0.31
CTSB P07858 2/20 0.31
CTSK P43235 2/20 0.31
CTSS P25774 1/20 0.31
KMT2A Q03164 1/20 0.31
MMP3 P08254 1/20 0.30
MMP9 P14780 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP3A4 P08684 1/20 0.30
CYP2C9 P11712 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7433589 0.88 MMP3 (0.36) MAOBALDH1A1POLBUSP2MAPT
SCHEMBL7433580 0.88 MMP3 (0.36) MAOBALDH1A1POLBUSP2MAPT
SCHEMBL7305075 0.87 CYP1A2 (0.42) ALDH1A1POLBUSP2MAPTHSD17B10
SCHEMBL7311340 0.87 POLB (0.40) ALDH1A1POLBUSP2MAPTHSD17B10
SCHEMBL7303801 0.86 ALDH1A1 (0.40) ALDH1A1POLBUSP2MAPTHSD17B10
SCHEMBL7434952 0.86 ALDH1A1 (0.35) ALDH1A1POLBUSP2MAPTHSD17B10
SCHEMBL8681390 0.85 CYP1A2 (0.36) ALDH1A1POLBUSP2MAPTHSD17B10
SCHEMBL7311350 0.85 TAS1R3 (0.38) ALDH1A1POLBUSP2MAPTHSD17B10
SCHEMBL7306052 0.84 ALDH1A1 (0.38) ALDH1A1POLBUSP2MAPTHSD17B10
SCHEMBL7311319 0.84 ALDH1A1 (0.37) ALDH1A1POLBUSP2MAPTHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0525420-B1 Pseudopeptides and dipeptides characterised by a substituted methyl ketone moiety at the C-terminus as thiol protease inhibitors MITSUBISHI CHEM CORP (JP) 1999-05-12 EP disclosed
US-5834508-A PROTEASE ENZYME INHIBITORS; MUSCLE DISORDERS MITSUBISHI CHEMICAL CORPORATION (JP) 1998-11-10 US disclosed
US-5639783-A POTENT PROTEASE INHIBITOR FOR TREATING MUSCULAR, NERVOUS SYSTEM DISEASES MITSUBISHI CHEMICAL CORPORATION (JP) 1997-06-17 US disclosed