SCHEMBL7433829

SCHEMBL7433829

CC(C)c1cc(NCc2ccc(-c3ccccc3-c3nnn[nH]3)cc2)n2nccc2n1

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KCNN3 Q9UGI6 3/20 0.45
KCNN1 Q92952 1/20 0.45
KCNN2 Q9H2S1 1/20 0.45
CCNT1 O60563 14/20 0.44
CDK9 P50750 14/20 0.44
CDK2 P24941 4/20 0.44
CCNE1 P24864 3/20 0.44
CDK4 P11802 3/20 0.44
CCND1 P24385 3/20 0.44
CDK1 P06493 1/20 0.44
CCNA2 P20248 1/20 0.44
CCNA1 P78396 1/20 0.44
CDK3 Q00526 1/20 0.44
CDK5 Q00535 1/20 0.44
CDK5R1 Q15078 1/20 0.44
CDK7 P50613 3/20 0.40
CCNH P51946 3/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7438720 0.88 KCNN3 (0.47) KCNN3KCNN1KCNN2CDK2CCNE1
SCHEMBL7441328 0.87 KCNN3 (0.62) KCNN3KCNN1KCNN2CDK2CCNE1
SCHEMBL7440984 0.86 AGTR1 (0.51) KCNN3KCNN1KCNN2CDK2CCNE1
SCHEMBL7438363 0.85 KCNN3 (0.45) KCNN3KCNN1KCNN2CDK2CCNE1
SCHEMBL7437203 0.85 KCNN3 (0.47) KCNN3KCNN1KCNN2CDK9CDK2
SCHEMBL7441634 0.84 KCNN3 (0.46) KCNN3KCNN1KCNN2CDK2CCNE1
SCHEMBL7438046 0.84 PDE10A (0.47) KCNN3KCNN1KCNN2CDK2CCNE1
SCHEMBL7442336 0.84 KCNN3 (0.45) KCNN3KCNN1KCNN2CDK2CCNE1
SCHEMBL7442662 0.83 KCNN3 (0.45) KCNN3KCNN1KCNN2CCNT1CDK9
SCHEMBL7439253 0.83 PDE7A (0.36) CCNT1CDK9CDK2CCNE1CDK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0628559-B1 Pyrimidine compounds and their use as pharmaceuticals BEIERSDORF LILLY GMBH (DE) 2002-04-03 EP disclosed
US-5602136-A Pyrimidine compounds and their use as pharmaceuticals BEIERSDORF-LILLY GMBH (DE) 1997-02-11 US disclosed
US-5602137-A Pyrimidine compounds and their use as pharmaceuticals BEIERSDORF-LILLY GMBH (DE) 1997-02-11 US disclosed
US-5571813-A Fused pyrimidine compounds and their use as pharmaceuticals BEIERSDORF-LILLY GMBH (DE) 1996-11-05 US disclosed
EP-0628559-A1 Pyrimidine compounds and their use as pharmaceuticals Beiersdorf-Lilly GmbH (DE) 1994-12-14 EP disclosed