SCHEMBL7439253

SCHEMBL7439253

CC(C)c1cc(SCc2ccc(-c3ccccc3-c3nnn[nH]3)cc2)n2nccc2n1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE7A Q13946 3/20 0.36
PDE7B Q9NP56 3/20 0.36
PDE4A P27815 3/20 0.36
PDE4B Q07343 3/20 0.36
PDE4C Q08493 3/20 0.36
PDE4D Q08499 3/20 0.36
PDE3B Q13370 3/20 0.36
PDE3A Q14432 3/20 0.36
CCNT1 O60563 13/20 0.36
CDK9 P50750 13/20 0.36
CDK4 P11802 3/20 0.36
CCND1 P24385 3/20 0.36
CDK1 P06493 1/20 0.36
CCNA2 P20248 1/20 0.36
CCNE1 P24864 1/20 0.36
CDK2 P24941 1/20 0.36
CCNA1 P78396 1/20 0.36
CDK3 Q00526 1/20 0.36
CDK5 Q00535 1/20 0.36
CDK5R1 Q15078 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7439761 0.88 UBE2M (0.38) PDE7APDE7BPDE4APDE4BPDE4C
SCHEMBL7435968 0.86 AGTR1 (0.36) PDE7APDE7BPDE4APDE4BPDE4C
SCHEMBL7443532 0.85 PDE4A (0.37) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL7437181 0.84 PKM (0.34) PDE7APDE7BPDE4APDE4BPDE4C
SCHEMBL7439344 0.84 PDE10A (0.31) PDE7APDE7BPDE4APDE4BPDE4C
SCHEMBL7439964 0.83 PDE4A (0.38) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL7433829 0.83 KCNN3 (0.45) CCNT1CDK9CDK4CCND1CDK1
SCHEMBL7433795 0.78 DPP4 (0.41) CCNT1CDK9CDK4CCND1CDK1
SCHEMBL7441634 0.73 KCNN3 (0.46) CCNE1CDK2
SCHEMBL7438720 0.72 KCNN3 (0.47) CCNE1CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0628559-B1 Pyrimidine compounds and their use as pharmaceuticals BEIERSDORF LILLY GMBH (DE) 2002-04-03 EP disclosed
US-5602137-A Pyrimidine compounds and their use as pharmaceuticals BEIERSDORF-LILLY GMBH (DE) 1997-02-11 US disclosed
US-5602136-A Pyrimidine compounds and their use as pharmaceuticals BEIERSDORF-LILLY GMBH (DE) 1997-02-11 US disclosed
US-5571813-A Fused pyrimidine compounds and their use as pharmaceuticals BEIERSDORF-LILLY GMBH (DE) 1996-11-05 US disclosed
EP-0628559-A1 Pyrimidine compounds and their use as pharmaceuticals Beiersdorf-Lilly GmbH (DE) 1994-12-14 EP disclosed