SCHEMBL7434130

SCHEMBL7434130

CC(C)[C](Cc1ccccc1)c1ccccc1C(C)C

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 3/20 0.41
GABRB2 P47870 2/20 0.41
TSHR P16473 2/20 0.41
GABRG2 P18507 2/20 0.38
GABRB3 P28472 2/20 0.38
CNR2 P34972 1/20 0.38
POLB P06746 2/20 0.38
SLC6A2 P23975 2/20 0.38
FAAH O00519 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
LMNA P02545 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
HPGD P15428 1/20 0.38
GABRB1 P18505 1/20 0.38
PTGS1 P23219 1/20 0.38
HTR2C P28335 1/20 0.38
GABRA5 P31644 1/20 0.38
GABRA3 P34903 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9131807 0.88 GABRA1 (0.41) GABRA1GABRB2TSHRGABRG2GABRB3
SCHEMBL9132471 0.86 TSHR (0.49) TSHRPOLBCES2CES1AKR1B1
SCHEMBL7430127 0.85 ALOX5 (0.50) SLC6A2LMNACYP1A2PTGS1HIF1A
SCHEMBL7444375 0.84 TRPA1 (0.39) GABRA1GABRB2TSHRGABRG2GABRB3
SCHEMBL9129189 0.82 HTR2A (0.46) CYP1A2HTR2CHTR2BCES2
SCHEMBL6547552 0.81 GABRA1 (0.41) GABRA1GABRB2TSHRGABRG2GABRB3
SCHEMBL9133864 0.79 GABRA1 (0.42) GABRA1GABRB2TSHRGABRG2GABRB3
SCHEMBL9129968 0.76 TSHR (0.46) TSHRCNR2POLBSLC6A2HPGD
SCHEMBL9130921 0.75 TSHR (0.47) TSHRPOLBCES2CES1AKR1B1
SCHEMBL9129992 0.75 ALDH1A1 (0.38) TSHRPOLBLMNAHPGDCES2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5491149-A VIRICIDES THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1996-02-13 US disclosed
US-5430155-A Viricides, treatment of AIDS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1995-07-04 US disclosed
US-5294720-A Viricides THE DUPONT MERCK PHARMACEUTICAL CO. (US) 1994-03-15 US disclosed
EP-0532693-A1 1,4-DIAMINO-2,3-DIHYDROXYBUTANES THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1993-03-24 EP disclosed