SCHEMBL762497

SCHEMBL762497

CC(C)(C)OC(=O)N1CCC[C@@H](c2nc3c(Cl)cccc3[nH]2)C1

nearest known ligand 0.52

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 10/20 0.52
HPGDS O60760 2/20 0.52
PTGES O14684 1/20 0.46
PTGS1 P23219 1/20 0.46
PTGS2 P35354 1/20 0.46
HCRTR1 O43613 2/20 0.45
HCRTR2 O43614 2/20 0.45
JAK2 O60674 1/20 0.44
JAK1 P23458 1/20 0.44
PRMT5 O14744 1/20 0.44
TRPV3 Q8NET8 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL743450 0.89 PTGS1 (0.57) PARP1HPGDSPTGS1PTGS2HCRTR1
SCHEMBL743449 0.89 PTGS1 (0.57) PARP1HPGDSPTGS1PTGS2HCRTR1
SCHEMBL20029041 0.88 PARP1 (0.52) PARP1HPGDSPTGS1PTGS2HCRTR1
SCHEMBL741851 0.87 PARP1 (0.51) PARP1HPGDSPTGS1PTGS2HCRTR1
SCHEMBL741850 0.87 PARP1 (0.51) PARP1HPGDSPTGS1PTGS2HCRTR1
SCHEMBL19951502 0.86 PARP1 (0.70) PARP1
SCHEMBL739293 0.84 PARP1 (0.54) PARP1PTGS1PTGS2HCRTR1HCRTR2
SCHEMBL742218 0.84 HPGDS (0.52) PARP1HPGDSJAK2JAK1PRMT5
SCHEMBL742219 0.84 HPGDS (0.52) PARP1HPGDSJAK2JAK1PRMT5
SCHEMBL739188 0.83 HPGDS (0.57) PARP1HPGDSPRMT5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed