SCHEMBL7436348

SCHEMBL7436348

COc1cc(N)c(Cl)cc1C(=O)NCC1CN2CCN1CC2

nearest known ligand 0.64

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTR4 Q13639 5/20 0.63
HTR3A P46098 4/20 0.63
DRD2 P14416 3/20 0.63
HTR3E A5X5Y0 2/20 0.63
HTR3B O95264 2/20 0.63
HTR3D Q70Z44 2/20 0.63
HTR3C Q8WXA8 2/20 0.63
DRD4 P21917 2/20 0.60
DRD3 P35462 2/20 0.60
HTR5A P47898 1/20 0.59
MEN1 O00255 1/20 0.59
CYP2D6 P10635 1/20 0.59
CYP2C9 P11712 1/20 0.59
CYP2C19 P33261 1/20 0.59
KMT2A Q03164 1/20 0.59
MAPK1 P28482 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8870896 0.99 HTR4 (0.62) HTR4HTR3ADRD2HTR3EHTR3B
SCHEMBL7433789 0.86 DRD2 (0.52) HTR4HTR3ADRD2HTR3EHTR3B
SCHEMBL7918548 0.82 HTR3A (0.69) HTR4HTR3ADRD2HTR3EHTR3B
SCHEMBL8854577 0.80 DRD2 (0.74) HTR4HTR3ADRD2HTR3EHTR3B
SCHEMBL11173712 0.78 HTR4 (0.65) HTR4HTR3ADRD2HTR3EHTR3B
SCHEMBL7354795 0.78 HTR4 (0.59) HTR4HTR3ADRD2HTR3EHTR3B
SCHEMBL7385997 0.78 DRD2 (0.75) HTR4DRD2DRD4DRD3
SCHEMBL10721765 0.78 HTR4 (0.64) HTR4HTR3ADRD2HTR3EHTR3B
SCHEMBL9021828 0.78 DRD2 (0.78) HTR4DRD2DRD4DRD3
SCHEMBL11179659 0.78 HTR4 (0.61) HTR4HTR3ADRD2HTR3EHTR3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0748807-A1 Derivatives of N-(1,4-diazabicyclo(2.2.2)-oct-2-yl)methyl benzamide, their preparation and their therapeutical use SYNTHELABO (FR) 1996-12-18 EP disclosed