SCHEMBL7437101

SCHEMBL7437101

c1ccc(CSC2(N3CCCCCC3)CCCCCC2)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 2/20 0.46
GRIN1 Q05586 2/20 0.46
GRIN2A Q12879 2/20 0.46
GRIN2B Q13224 2/20 0.46
SLC6A3 Q01959 2/20 0.46
GRIN2D O15399 1/20 0.46
GRIN3B O60391 1/20 0.46
CYP2B6 P20813 1/20 0.46
SLC6A2 P23975 1/20 0.46
SLC6A4 P31645 1/20 0.46
PRCP P42785 1/20 0.46
KCNH2 Q12809 1/20 0.46
GRIN2C Q14957 1/20 0.46
GRIN3A Q8TCU5 1/20 0.46
OPRM1 P35372 1/20 0.45
OPRD1 P41143 1/20 0.45
TSHR P16473 2/20 0.40
MEN1 O00255 3/20 0.38
KMT2A Q03164 3/20 0.38
HTT P42858 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11619698 0.76 KMT2A (0.42) SLC6A4MEN1KMT2AHTTHPGD
SCHEMBL11066307 0.74 SIGMAR1 (0.50) SIGMAR1GRIN1GRIN2AGRIN2BSLC6A3
SCHEMBL27174624 0.73 IDO1 (0.39) SLC6A4MEN1KMT2AHTT
SCHEMBL29093049 0.71 IDO1 (0.41) MEN1KMT2AHTTHPGD
SCHEMBL8635453 0.70 SIGMAR1 (0.50) SIGMAR1GRIN1GRIN2AGRIN2BSLC6A3
SCHEMBL3404247 0.69 DPP4 (0.43) SLC6A3SLC6A2SLC6A4MEN1KMT2A
SCHEMBL18429033 0.69 SIGMAR1 (0.48) SIGMAR1SLC6A3TSHRMEN1KMT2A
Hydrochloric Acid SCHEMBL29424738 0.67 SIGMAR1 (0.47) SIGMAR1SLC6A3TSHRMEN1KMT2A
SCHEMBL1983726 0.66 CYP2C19 (0.41) TSHRMEN1KMT2AHPGDGAA
SCHEMBL7323247 0.66 ALDH1A1 (0.36) SLC6A4TSHRMEN1KMT2AHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0710237-A1 QUINOLIZIDINES WITH CALCIUM CHANNEL ANTAGONISTIC ACTIVITY SMITHKLINE BEECHAM PLC (GB) 1996-05-08 EP disclosed
WO-1995003302-A1 QUINOLIZIDINES WITH CALCIUM CHANNEL ANTAGONISTIC ACTIVITY SMITHKLINE BEECHAM PLC (GB) 1995-02-02 WO disclosed