SCHEMBL7437388

SCHEMBL7437388

CCCCn1c(=O)c(O)c(C(=O)O)c2ccccc21

nearest known ligand 0.68

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.66
MEN1 O00255 5/20 0.63
KMT2A Q03164 5/20 0.63
SMN1; SMN2 Q16637 2/20 0.63
KDM4E B2RXH2 6/20 0.62
LMNA P02545 3/20 0.62
HPGD P15428 3/20 0.62
POLB P06746 1/20 0.62
PGR P06401 1/20 0.61
RORA P35398 1/20 0.61
RORC P51449 1/20 0.61
RORB Q92753 1/20 0.61
MAPT P10636 1/20 0.60
HTT P42858 3/20 0.57
TP53 P04637 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27854528 0.89 MEN1 (0.74) ALDH1A1MEN1KMT2ASMN1; SMN2KDM4E
SCHEMBL7435666 0.85 KDM4E (0.61) ALDH1A1MEN1KMT2ASMN1; SMN2KDM4E
SCHEMBL29280449 0.85 MEN1 (0.74) ALDH1A1MEN1KMT2ASMN1; SMN2KDM4E
SCHEMBL6126717 0.84 HTT (0.74) ALDH1A1MEN1KMT2ASMN1; SMN2KDM4E
SCHEMBL27854540 0.83 L3MBTL1 (0.69) ALDH1A1MEN1KMT2ASMN1; SMN2KDM4E
SCHEMBL8784179 0.81 AGTR1 (0.55) ALDH1A1MEN1KMT2ASMN1; SMN2KDM4E
Hydrochloric Acid SCHEMBL7348525 0.80 CNR2 (0.52) ALDH1A1KDM4EHPGDPOLBPGR
Hydrochloric Acid SCHEMBL7347698 0.80 CNR2 (0.55) ALDH1A1KDM4EHPGDPOLBPGR
SCHEMBL9591254 0.79 KDM4E (0.76) ALDH1A1MEN1KMT2ASMN1; SMN2KDM4E
SCHEMBL7437202 0.78 ALDH1A1 (0.62) ALDH1A1MEN1KMT2ASMN1; SMN2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0458636-B1 Antiemetic and migraine suppressing heterocyclic compounds and pharmaceutical compositions containing them KYOWA HAKKO KOGYO KK (JP) 1995-07-12 EP disclosed
US-5248684-A CERTAIN 2-OXO-QUINOLINE CARBOXYLATES OR CORRESPONDING CARBOXAMIDES USEFUL AS ANTI-EMETICS AND SUPPRESSANTS OF MIGRAINE KYOWA HAKKO KOGYO CO., LTD. (JP) 1993-09-28 US disclosed
EP-0458636-A1 Antiemetic and migraine suppressing heterocyclic compounds and pharmaceutical compositions containing them KYOWA HAKKO KOGYO CO., LTD (JP) 1991-11-27 EP disclosed