SCHEMBL7438151

SCHEMBL7438151

C=CC[C@@H](Nc1ccccc1)c1ccc(C)cc1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.50
ALDH1A1 P00352 4/20 0.50
KDM4E B2RXH2 1/20 0.50
ALOX15 P16050 1/20 0.50
HSD17B10 Q99714 1/20 0.50
SMN1; SMN2 Q16637 2/20 0.47
ATM Q13315 2/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
NPBWR1 P48145 1/20 0.44
MCHR1 Q99705 1/20 0.44
VDR P11473 1/20 0.43
TP53 P04637 3/20 0.41
CYP2C19 P33261 3/20 0.41
NPSR1 Q6W5P4 2/20 0.41
GAA P10253 2/20 0.41
CYP1A2 P05177 2/20 0.41
CYP3A4 P08684 2/20 0.41
CYP2D6 P10635 2/20 0.41
MEN1 O00255 1/20 0.41
LMNA P02545 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7438162 0.94 ALDH1A1 (0.54) MAPTALDH1A1KDM4EALOX15HSD17B10
SCHEMBL14457019 0.88 ALDH1A1 (0.61) MAPTALDH1A1KDM4EALOX15HSD17B10
SCHEMBL29741303 0.78 TEAD4 (0.47) MAPTALDH1A1ALOX15SMN1; SMN2ATM
SCHEMBL15787624 0.78 SMN1; SMN2 (0.42) MAPTALDH1A1KDM4EALOX15HSD17B10
SCHEMBL15787285 0.78 SMN1; SMN2 (0.42) MAPTALDH1A1KDM4EALOX15HSD17B10
SCHEMBL13675544 0.77 MAPT (0.50) MAPTALDH1A1ALOX15SMN1; SMN2ATM
SCHEMBL13675806 0.77 MAPT (0.50) MAPTALDH1A1ALOX15SMN1; SMN2ATM
SCHEMBL16521856 0.75 CYP3A4 (0.44) MAPTALDH1A1KDM4EALOX15HSD17B10
SCHEMBL5512077 0.73 VDR (0.58) MAPTALDH1A1ALOX15SMN1; SMN2NPBWR1
SCHEMBL31147708 0.73 NPBWR1 (0.43) MAPTALDH1A1ALOX15SMN1; SMN2ATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5229381-A Inhibitors of leukocyte enzyme elastase MERCK & CO., INC. (US) 1993-07-20 US disclosed
EP-0481671-A1 New substituted azetidinones as anti-inflammatory and antidegenerative agents MERCK & CO. INC. (US) 1992-04-22 EP disclosed