SCHEMBL7439002

SCHEMBL7439002

CC(C)C[C@H](Nc1nc(-c2cccc(NC(=O)NCCc3ccccc3)c2)cs1)C(=O)NCC#N

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 1/20 0.50
ROCK1 Q13464 1/20 0.50
MAPT P10636 6/20 0.47
KDM4E B2RXH2 2/20 0.47
ALDH1A1 P00352 2/20 0.47
SMN1; SMN2 Q16637 3/20 0.47
HTT P42858 2/20 0.47
MEN1 O00255 5/20 0.47
KMT2A Q03164 5/20 0.47
TP53 P04637 1/20 0.47
ANPEP P15144 1/20 0.45
CTSK P43235 4/20 0.45
LMNA P02545 1/20 0.43
CTSS P25774 5/20 0.43
CTSL P07711 4/20 0.43
CTSB P07858 3/20 0.43
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
MRE11 P49959 1/20 0.43
MAPK1 P28482 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6185021 0.91 MEN1 (0.52) ROCK1MAPTKDM4EALDH1A1SMN1; SMN2
SCHEMBL6180437 0.87 ROCK2 (0.50) ROCK2ROCK1MAPTKDM4EALDH1A1
SCHEMBL6181829 0.85 MEN1 (0.52) MAPTKDM4EALDH1A1SMN1; SMN2HTT
SCHEMBL6180116 0.83 CTSK (0.56) MEN1KMT2ACTSKCTSSCTSL
SCHEMBL6183760 0.80 CTSL (0.49) CTSKCTSSCTSLCTSB
SCHEMBL6181675 0.80 HDAC3 (0.44) MAPTKDM4EALDH1A1SMN1; SMN2HTT
SCHEMBL7433934 0.79 MAPT (0.58) ROCK1MAPTKDM4EALDH1A1SMN1; SMN2
SCHEMBL7433950 0.79 MAPT (0.58) ROCK1MAPTKDM4EALDH1A1SMN1; SMN2
SCHEMBL7651961 0.79 CTSS (0.47) MAPTKDM4EALDH1A1SMN1; SMN2HTT
SCHEMBL6181689 0.79 CTSS (0.47) MAPTKDM4EALDH1A1SMN1; SMN2HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001068645-A2 N-CYANOMETHYLCARBOXAMIDES AND THEIR USE AS PROTEASE INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2001-09-20 WO claimed
WO-2001068645-A2 N-CYANOMETHYLCARBOXAMIDES AND THEIR USE AS PROTEASE INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2001-09-20 WO disclosed