SCHEMBL7439103

SCHEMBL7439103

CC(=O)SCC(Cc1ccccc1)NC(=O)C(Cc1ccc(-c2ccccc2)c(C#N)c1)C(=O)O

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MME P08473 5/20 0.43
ITGB1 P05556 1/20 0.42
ITGA4 P13612 1/20 0.42
FCER2 P06734 1/20 0.40
PTPN1 P18031 1/20 0.40
CTSS P25774 2/20 0.39
CTSK P43235 1/20 0.39
CYP3A4 P08684 1/20 0.39
MAPK1 P28482 1/20 0.39
MRE11 P49959 1/20 0.39
CTSL P07711 1/20 0.38
CTSB P07858 1/20 0.38
ACE P12821 3/20 0.38
CPA1 P15085 2/20 0.37
ACE2 Q9BYF1 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7450894 0.82 MME (0.52) MMEFCER2CYP3A4MAPK1ACE
SCHEMBL7609959 0.76 MME (0.57) MMEITGB1ITGA4PTPN1ACE
SCHEMBL20474596 0.74 CTSC (0.48) MMEITGB1ITGA4PTPN1CTSK
SCHEMBL18554154 0.74 CTSC (0.48) MMEITGB1ITGA4PTPN1CTSK
SCHEMBL4018176 0.73 SLC22A12 (0.42) MMEITGB1ITGA4PTPN1MRE11
SCHEMBL4018178 0.73 SLC22A12 (0.42) MMEITGB1ITGA4PTPN1MRE11
SCHEMBL27792670 0.72 MMP8 (0.46)
SCHEMBL4448448 0.72 CYP19A1 (0.41) MMEITGB1ITGA4PTPN1MRE11
SCHEMBL8837469 0.70 FCER2 (0.50) MMEFCER2CYP3A4MAPK1ACE
SCHEMBL3178122 0.69 CYP19A1 (0.51) MMECTSSCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0888299-A1 SULPHUR DERIVATIVES WITH A RETROAMIDE BOND AS ENDOTHELIN-CONVERTING ENZYME INHIBITORS HOECHST MARION ROUSSEL (FR) 1999-01-07 EP disclosed
WO-1997032849-A1 SULPHUR DERIVATIVES WITH A RETROAMIDE BOND AS ENDOTHELIN-CONVERTING ENZYME INHIBITORS HOECHST MARION ROUSSEL (FR) 1997-09-12 WO disclosed