SCHEMBL7439629

SCHEMBL7439629

O=C(NCc1ccc(S(=O)(=O)N2CCN(CCc3ccccc3)CC2)s1)c1ccc(Cl)cc1.O=C(NCc1ccc(S(=O)(=O)N2CCN(Cc3ccc(F)cc3)CC2)s1)c1ccc(Cl)cc1

nearest known ligand 0.51

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MAPK9 P45984 1/20 0.51
MAPK10 P53779 1/20 0.51
BCL2 P10415 1/20 0.49
BCL2L1 Q07817 1/20 0.49
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
LMNA P02545 2/20 0.48
SMN1; SMN2 Q16637 2/20 0.48
MAPK1 P28482 1/20 0.48
ALDH1A1 P00352 2/20 0.45
PRKAA2 P54646 2/20 0.45
GLS O94925 1/20 0.44
CHRM4 P08173 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6431959 0.95 MAPK9 (0.55) MAPK9MAPK10BCL2BCL2L1MEN1
SCHEMBL3479899 0.93 MAPK9 (0.57) MAPK9MAPK10BCL2BCL2L1MEN1
SCHEMBL3480113 0.92 MAPK9 (0.54) MAPK9MAPK10BCL2BCL2L1MEN1
SCHEMBL3480648 0.90 MAPK9 (0.60) MAPK9MAPK10BCL2BCL2L1MEN1
SCHEMBL2423789 0.88 MAPK9 (0.56) MAPK9MAPK10BCL2BCL2L1MEN1
SCHEMBL7440295 0.84 DRD2 (0.54) MAPK9MAPK10BCL2BCL2L1MEN1
SCHEMBL2426839 0.81 MEN1 (0.53) MAPK9MAPK10BCL2BCL2L1MEN1
SCHEMBL2421342 0.81 MAPK9 (0.56) MAPK9MAPK10BCL2BCL2L1MEN1
SCHEMBL7434542 0.81 DRD2 (0.58) MAPK9MAPK10BCL2BCL2L1MEN1
SCHEMBL7704876 0.81 ALDH1A1 (0.57) MAPK9MAPK10BCL2BCL2L1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1218374-A1 PHARMACEUTICALLY ACTIVE SULFONAMIDE DERIVATIVES Applied Research Systems ARS Holding N.V. (AN) 2002-07-03 EP claimed
WO-2001023378-A1 PHARMACEUTICALLY ACTIVE SULFONAMIDE DERIVATIVES APPLIED RESEARCH SYSTEMS ARS HOLDING N.V. (AN) 2001-04-05 WO claimed