SCHEMBL7441589

SCHEMBL7441589

CCOC(=O)Cc1ccc(OCCCN2CCC(C(c3ccc(F)cc3)c3ccc(F)c(F)c3)CC2)c(OC)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.41
ALDH1A1 P00352 1/20 0.41
MAPK1 P28482 1/20 0.41
ACHE P22303 3/20 0.41
HTR1A P08908 4/20 0.40
DRD2 P14416 4/20 0.40
HTR2A P28223 4/20 0.40
HRH3 Q9Y5N1 3/20 0.40
CHRM1 P11229 2/20 0.40
CHRM4 P08173 1/20 0.40
CHRM5 P08912 1/20 0.40
ABCB11 O95342 1/20 0.40
CHRM2 P08172 1/20 0.40
ADRA2A P08913 1/20 0.40
ADRA2B P18089 1/20 0.40
ADRA2C P18825 1/20 0.40
DRD1 P21728 1/20 0.40
DRD4 P21917 1/20 0.40
SLC6A2 P23975 1/20 0.40
HTR2C P28335 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7443381 0.88 DRD2 (0.44) KDM4EALDH1A1MAPK1ACHEHTR1A
SCHEMBL7433713 0.86 HTR1A (0.43) KDM4EALDH1A1MAPK1ACHEHTR1A
SCHEMBL7443763 0.86 KCNH2 (0.44) KDM4EALDH1A1MAPK1HTR1ADRD2
SCHEMBL10460769 0.85 ABCB11 (0.56) KDM4EALDH1A1ACHEHTR1ADRD2
SCHEMBL7441777 0.84 KCNH2 (0.48) ACHEHTR1ADRD2HTR2ACHRM1
SCHEMBL7446532 0.83 ABCB11 (0.47) KDM4EALDH1A1ACHEHTR1ADRD2
Oxalic Acid SCHEMBL10460714 0.83 KDM4E (0.53) KDM4EALDH1A1MAPK1ACHEHTR1A
Oxalic Acid SCHEMBL10461465 0.83 ABCB11 (0.54) KDM4EALDH1A1ACHEHTR1ADRD2
SCHEMBL7437606 0.82 ABCB11 (0.47) KDM4EALDH1A1ACHEHTR1ADRD2
SCHEMBL10461677 0.82 KDM4E (0.49) KDM4EALDH1A1MAPK1HTR1ADRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5070087-A Aryl(alkyland alkylene)-N-((phenoxy and phenylthio)alkyl) aminoheterocyclics as cardiovascular, anthihistaminic, antisecretory and antiallergy agents A. H. ROBINS COMPANY, INCORPORATED (US) 1991-12-03 US disclosed