SCHEMBL7443203

SCHEMBL7443203

C[C@H](NC(=O)C(=O)C(CC(F)(F)F)NC(=O)OC(C)(C)C)c1ccc2ccccc2c1

nearest known ligand 0.55

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CTSK P43235 13/20 0.55
MMP9 P14780 1/20 0.50
GABRB1 P18505 1/20 0.48
GABRB2 P47870 1/20 0.48
CTSB P07858 2/20 0.46
CTSS P25774 2/20 0.46
CTSL P07711 1/20 0.40
CTSH P09668 1/20 0.40
PTPN1 P18031 1/20 0.40
HCRTR1 O43613 1/20 0.40
TDP1 Q9NUW8 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7442582 0.88 CTSK (0.46) CTSKGABRB1GABRB2CTSBCTSS
SCHEMBL7437012 0.87 CTSK (0.71) CTSKCTSBCTSSCTSLCTSH
SCHEMBL13715427 0.82 MMP9 (0.59) CTSKMMP9GABRB1GABRB2CTSB
SCHEMBL7430555 0.81 METAP2 (0.47) CTSKMMP9GABRB1GABRB2CTSB
SCHEMBL7446907 0.79 CTSK (0.56) CTSKGABRB1GABRB2CTSBCTSS
SCHEMBL7447101 0.79 CTSK (0.56) CTSKGABRB1GABRB2CTSBCTSS
SCHEMBL7447637 0.79 CTSK (0.52) CTSKGABRB1GABRB2CTSBCTSS
SCHEMBL7439368 0.77 CTSK (0.56) CTSKGABRB1GABRB2CTSBCTSS
SCHEMBL7430637 0.77 CTSK (0.56) CTSKGABRB1GABRB2CTSBCTSS
SCHEMBL7443211 0.77 MMP9 (0.47) CTSKMMP9GABRB1GABRB2HCRTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6187905-B1 PEPTIDE COMPOUND WHICH INHIBITS VIRAL PROTEINASES; VIRICIDES FOR HEPATITIS C, HEPATITIS G, AND HUMAN GB VIRUSES HOFFMANN-LA ROCHE INC. 2001-02-13 US disclosed