SCHEMBL7444588

SCHEMBL7444588

N#Cc1ccc(C(=O)CC2C=COc3ccccc32)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 2/20 0.43
SIGMAR1 Q99720 1/20 0.41
POLB P06746 1/20 0.41
CA1 P00915 2/20 0.36
CA2 P00918 2/20 0.36
ALDH1A1 P00352 2/20 0.36
LMNA P02545 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
RAB9A P51151 1/20 0.35
MEN1 O00255 1/20 0.35
NPC1 O15118 1/20 0.35
KMT2A Q03164 1/20 0.35
HTR1A P08908 1/20 0.35
DRD2 P14416 1/20 0.35
HTR2A P28223 1/20 0.35
SLC6A4 P31645 1/20 0.35
HTR7 P34969 1/20 0.35
HRH1 P35367 1/20 0.35
DRD3 P35462 1/20 0.35
HTR2B P41595 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8389861 0.80 MAPK1 (0.42) POLBALDH1A1MEN1KMT2AMAPK1
SCHEMBL1574529 0.76 EGFR (0.36) ALDH1A1LMNAMEN1KMT2AMAPK1
SCHEMBL3430197 0.75 ATM (0.41) LMNAMEN1KMT2AMAPK1
SCHEMBL12700339 0.70 LMNA (0.58) GSK3BSIGMAR1POLBALDH1A1LMNA
SCHEMBL8309737 0.70 IDO1 (0.35) MEN1KMT2A
SCHEMBL7439230 0.69 GSK3B (0.46) GSK3BSIGMAR1POLBCA1CA2
SCHEMBL16088741 0.67 HSD17B10 (0.57) GSK3BSIGMAR1POLBCA1CA2
SCHEMBL28043310 0.66 KMT2A (0.65) GSK3BPOLBCA1CA2ALDH1A1
SCHEMBL9772861 0.66 HTR2A (0.36) MEN1KMT2AHTR2ASLC6A4HRH1
SCHEMBL293418 0.66 MAOA (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0849263-A2 Pharmaceutical substituted propanoic acid derivatives ELI LILLY AND COMPANY LIMITED (GB) 1998-06-24 EP disclosed