SCHEMBL7445085

SCHEMBL7445085

C[C@@H](C(=O)O)N(C(=O)CCN1CCOCC1)c1ccccc1

nearest known ligand 0.56

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.56
MAPT P10636 2/20 0.56
KMT2A Q03164 2/20 0.56
LMNA P02545 2/20 0.49
CYP2C19 P33261 1/20 0.49
HSP90AA1 P07900 1/20 0.46
OPRM1 P35372 1/20 0.46
OPRD1 P41143 1/20 0.46
NPC1 O15118 1/20 0.45
KDM4E B2RXH2 1/20 0.44
GAA P10253 1/20 0.44
GLA P06280 1/20 0.43
TERT O14746 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7297001 0.87 ALDH1A1 (0.53) ALDH1A1MAPTKMT2ALMNANPC1
SCHEMBL7445245 0.79 ALDH1A1 (0.57) ALDH1A1KMT2ALMNACYP2C19GAA
SCHEMBL31479993 0.76 ALDH1A1 (0.51) ALDH1A1KMT2ALMNAOPRD1GAA
SCHEMBL27615561 0.76 ALDH1A1 (0.45) ALDH1A1KMT2ALMNA
SCHEMBL11272120 0.74 ALDH1A1 (0.49) ALDH1A1KMT2ALMNANPC1GLA
SCHEMBL8922653 0.73 ALDH1A1 (0.54) ALDH1A1MAPTKMT2ALMNAOPRM1
SCHEMBL7445267 0.73 MLYCD (0.55) ALDH1A1KMT2ALMNAOPRM1OPRD1
SCHEMBL321369 0.72 ALDH1A1 (1.00) ALDH1A1MAPTKMT2ALMNACYP2C19
SCHEMBL22858397 0.72 ALDH1A1 (0.55) ALDH1A1MAPTKMT2ALMNACYP2C19
SCHEMBL20421705 0.72 ALDH1A1 (0.53) ALDH1A1KMT2ALMNANPC1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0817795-B1 NOVEL 4-SUBSTITUTED-3-PEPTIDYL-AZETIDIN-2-ONE DERIVATIVES USEFUL AS CYSTEINE PROTEINASE INHIBITOR NAEJA PHARMACEUTICAL INC (CA) 2000-11-15 EP disclosed
US-5986108-A ENZYME INHIBITORS SYNPHAR LABORATORIES, INC. (CA) 1999-11-16 US disclosed
EP-0817795-A1 NOVEL 4-SUBSTITUTED-3-PEPTIDYL-AZETIDIN-2-ONE DERIVATIVES USEFUL AS CYSTEINE PROTEINASE INHIBITOR SYNPHAR LABORATORIES INC. (CA) 1998-01-14 EP disclosed
WO-1996032408-A1 NOVEL 4-SUBSTITUTED-3-PEPTIDYL-AZETIDIN-2-ONE DERIVATIVES USEFUL AS CYSTEINE PROTEINASE INHIBITOR SYNPHAR LABORATORIES, INC. (US) 1996-10-17 WO disclosed