SCHEMBL7445238

SCHEMBL7445238

CCCN(CCC)C1Cc2cc3[nH]cc(C(=O)CC)c3cc2C1

nearest known ligand 0.55

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 1/20 0.50
HTR1D P28221 6/20 0.49
FYN P06241 1/20 0.49
HTR1B P28222 5/20 0.45
DRD2 P14416 2/20 0.45
ALDH1A1 P00352 2/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C9 P11712 1/20 0.44
ALOX15 P16050 1/20 0.44
MAPK1 P28482 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7445106 0.92 HTR1D (0.57) HTR1AHTR1DFYNHTR1BDRD2
SCHEMBL7438442 0.91 HTR1A (0.46) HTR1AHTR1DFYNHTR1BDRD2
SCHEMBL7439655 0.83 HTR1A (0.48) HTR1AHTR1DFYNHTR1BDRD2
SCHEMBL7443429 0.78 HTR1D (0.53) HTR1AHTR1DFYNHTR1BALDH1A1
SCHEMBL7208944 0.75 HTR1A (0.81) HTR1AHTR1DHTR1BDRD2
SCHEMBL7444866 0.74 HTR1A (0.41) HTR1AHTR1DHTR1BDRD2
SCHEMBL7441439 0.73 HTR1D (0.69) HTR1AHTR1DHTR1BDRD2
SCHEMBL7460946 0.71 FYN (0.65) HTR1AFYNDRD2ALDH1A1CYP2D6
SCHEMBL7445758 0.71 HTR1D (0.62) HTR1AHTR1DFYNHTR1B
SCHEMBL7439653 0.71 HTR1B (0.46) HTR1AHTR1DFYNHTR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5639778-A TREATING CENTRAL NERVOUS SYSTEM DISORDERS PHARMACIA & UPJOHN COMPANY (US) 1997-06-17 US disclosed
EP-0690843-A1 INDOLETETRALINS HAVING DOPAMINERGIC ACTIVITY PHARMACIA & UPJOHN COMPANY (US) 1996-01-10 EP disclosed
WO-1994021608-A1 INDOLETETRALINS HAVING DOPAMINERGIC ACTIVITY THE UPJOHN COMPANY (US) 1994-09-29 WO disclosed