SCHEMBL7445643

SCHEMBL7445643

CCOC(=O)C(NCC(C)(C(=O)N1CCCC1)c1ccc2[nH]c(CNc3ccc(C#N)cc3)nc2c1C)C(C)=O

nearest known ligand 0.35

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.35
ALDH1A1 P00352 1/20 0.35
LMNA P02545 1/20 0.35
MAPT P10636 1/20 0.35
MAPK1 P28482 1/20 0.35
RAB9A P51151 1/20 0.35
P2RY12 Q9H244 1/20 0.32
MLLT1 Q03111 1/20 0.32
DGAT2 Q96PD7 1/20 0.31
PIP4K2A P48426 1/20 0.31
TGFBR1 P36897 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7447916 0.88 RAB9A (0.38) NPC1ALDH1A1LMNAMAPTMAPK1
Hydrochloric Acid SCHEMBL7451196 0.88 RAB9A (0.38) NPC1ALDH1A1LMNAMAPTMAPK1
SCHEMBL7447469 0.85 NPC1 (0.36) NPC1ALDH1A1LMNAMAPTMAPK1
SCHEMBL7452254 0.85 RAB9A (0.38) NPC1ALDH1A1LMNAMAPTMAPK1
SCHEMBL7449208 0.85 NPC1 (0.39) NPC1ALDH1A1LMNAMAPTMAPK1
SCHEMBL7421109 0.84 NPC1 (0.37) NPC1ALDH1A1LMNAMAPTMAPK1
SCHEMBL7447757 0.83 NPC1 (0.34) NPC1ALDH1A1LMNAMAPTMAPK1
SCHEMBL7449699 0.82 MLLT1 (0.38) NPC1ALDH1A1LMNAMAPTMAPK1
SCHEMBL7446035 0.81 NPC1 (0.34) NPC1ALDH1A1LMNAMAPTMAPK1
SCHEMBL7454489 0.81 NPC1 (0.38) NPC1ALDH1A1LMNAMAPTMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1095025-A2 BENZIMIDAZOLES, PRODUCTION THEREOF AND USE THEREOF AS MEDICAMENTS BOEHRINGER INGELHEIM KG (DE) 2001-05-02 EP disclosed
WO-2000001704-A2 BENZIMIDAZOLES, PRODUCTION THEREOF AND USE THEREOF AS MEDICAMENTS BOEHRINGER INGELHEIM PHARMA KG (DE) 2000-01-13 WO disclosed