SCHEMBL7446035

SCHEMBL7446035

CCCCOC(=O)NC(=N)c1ccc(NCc2nc3c(C)c(C(C)(CNC(C(C)=O)C(=O)OC)C(=O)N4CCCC4)ccc3[nH]2)cc1

nearest known ligand 0.34

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.34
RAB9A P51151 3/20 0.34
MAPT P10636 2/20 0.34
ALDH1A1 P00352 1/20 0.34
LMNA P02545 1/20 0.34
MAPK1 P28482 1/20 0.34
KLK1 P06870 1/20 0.30
KLK5 Q9Y337 1/20 0.30
F2 P00734 1/20 0.30
F10 P00742 1/20 0.30
CASP1 P29466 1/20 0.30
TP53 P04637 1/20 0.30
NFKB1 P19838 1/20 0.30
NFKB2 Q00653 1/20 0.30
KMT2A Q03164 1/20 0.30
RELA Q04206 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7446732 0.97 NPC1 (0.33) NPC1RAB9AMAPTALDH1A1LMNA
SCHEMBL7447757 0.94 NPC1 (0.34) NPC1RAB9AMAPTALDH1A1LMNA
SCHEMBL7452254 0.94 RAB9A (0.38) NPC1RAB9AMAPTALDH1A1LMNA
SCHEMBL7447916 0.92 RAB9A (0.38) NPC1RAB9AMAPTALDH1A1LMNA
SCHEMBL7451026 0.89 ALDH1A1 (0.36) NPC1RAB9AMAPTALDH1A1LMNA
SCHEMBL7447469 0.88 NPC1 (0.36) NPC1RAB9AMAPTALDH1A1LMNA
SCHEMBL7449208 0.86 NPC1 (0.39) NPC1RAB9AMAPTALDH1A1LMNA
Hydrochloric Acid SCHEMBL7451196 0.84 RAB9A (0.38) NPC1RAB9AMAPTALDH1A1LMNA
SCHEMBL7446181 0.83 RAB9A (0.37) NPC1RAB9AMAPTALDH1A1LMNA
SCHEMBL7452478 0.82 F2 (0.36) NPC1RAB9AMAPTALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1095025-A2 BENZIMIDAZOLES, PRODUCTION THEREOF AND USE THEREOF AS MEDICAMENTS BOEHRINGER INGELHEIM KG (DE) 2001-05-02 EP disclosed
WO-2000001704-A2 BENZIMIDAZOLES, PRODUCTION THEREOF AND USE THEREOF AS MEDICAMENTS BOEHRINGER INGELHEIM PHARMA KG (DE) 2000-01-13 WO disclosed