SCHEMBL7449699

SCHEMBL7449699

Cc1c([C@@](C)(N)C(=O)N2CCCC2)ccc2[nH]c(CNc3ccc(C#N)cc3)nc12

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MLLT1 Q03111 1/20 0.38
DGAT2 Q96PD7 2/20 0.36
IDH1 O75874 2/20 0.35
TGFBR1 P36897 4/20 0.35
NPC1 O15118 1/20 0.35
ALDH1A1 P00352 1/20 0.35
LMNA P02545 1/20 0.35
MAPT P10636 1/20 0.35
MAPK1 P28482 1/20 0.35
RAB9A P51151 1/20 0.35
OPRM1 P35372 1/20 0.34
CSNK1E P49674 1/20 0.33
F2 P00734 1/20 0.33
F10 P00742 1/20 0.33
KLK1 P06870 2/20 0.33
KLK5 Q9Y337 2/20 0.33
MAPK14 Q16539 1/20 0.33
DPP7 Q9UHL4 1/20 0.32
PDK1 Q15118 1/20 0.32
PDK2 Q15119 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7442673 0.85 MLLT1 (0.34) MLLT1DGAT2IDH1TGFBR1NPC1
SCHEMBL7454489 0.83 NPC1 (0.38) MLLT1DGAT2IDH1TGFBR1NPC1
SCHEMBL7446445 0.83 NPC1 (0.38) MLLT1DGAT2IDH1TGFBR1NPC1
SCHEMBL7447136 0.83 ALDH1A1 (0.37) MLLT1DGAT2IDH1TGFBR1NPC1
SCHEMBL7410290 0.83 JAK2 (0.36) NPC1ALDH1A1LMNAMAPTMAPK1
SCHEMBL7421109 0.82 NPC1 (0.37) MLLT1DGAT2IDH1TGFBR1NPC1
SCHEMBL7445643 0.82 NPC1 (0.35) MLLT1DGAT2TGFBR1NPC1ALDH1A1
SCHEMBL7447505 0.82 NPC1 (0.36) MLLT1DGAT2IDH1TGFBR1NPC1
SCHEMBL7448201 0.81 EPHX2 (0.39) MLLT1DGAT2IDH1TGFBR1NPC1
SCHEMBL6457217 0.75 F2 (0.56) NPC1ALDH1A1LMNAMAPTMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1095025-A2 BENZIMIDAZOLES, PRODUCTION THEREOF AND USE THEREOF AS MEDICAMENTS BOEHRINGER INGELHEIM KG (DE) 2001-05-02 EP disclosed
WO-2000001704-A2 BENZIMIDAZOLES, PRODUCTION THEREOF AND USE THEREOF AS MEDICAMENTS BOEHRINGER INGELHEIM PHARMA KG (DE) 2000-01-13 WO disclosed